SCHEMBL30948977

SCHEMBL30948977

Cc1nc(Cl)ccc1-c1ncn(C)n1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 6/20 0.39
HCRTR2 O43614 6/20 0.39
MC4R P32245 1/20 0.37
PPARA Q07869 1/20 0.34
AXL P30530 2/20 0.31
GABRG2 P18507 1/20 0.30
GABRB3 P28472 1/20 0.30
GABRA5 P31644 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30948975 0.75 NR1H2 (0.34) AXL
SCHEMBL30996534 0.73 EPHX2 (0.37) PPARA
SCHEMBL30833320 0.73 TDP1 (0.37)
SCHEMBL23837827 0.70 IDO1 (0.41) HCRTR1HCRTR2
SCHEMBL25435848 0.70 LRRK2 (0.41) HCRTR1HCRTR2
SCHEMBL2276312 0.69 CHRNB2 (0.43) PPARA
SCHEMBL31634725 0.69 MC4R (0.37) MC4R
SCHEMBL20969942 0.69 PPARA (0.40) PPARAGABRG2GABRB3GABRA5
SCHEMBL12331975 0.68 PPARA (0.37) HCRTR1HCRTR2PPARA
SCHEMBL31646940 0.68 BRD4 (0.43) HCRTR1HCRTR2MC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4620955-A1 MC4R ANTAGONIST COMPOUND, PHARMACEUTICAL COMPOSITION AND PHARMACEUTICAL USE THEREOF Changchun Genescience Pharmaceutical Co., Ltd. (CN) 2025-09-24 EP disclosed
CN-120202199-A MC4R antagonist compound, pharmaceutical composition and application thereof in medicine 长春金赛药业有限责任公司 2025-06-24 CN disclosed
WO-2024104452-A1 MC4R ANTAGONIST COMPOUND, PHARMACEUTICAL COMPOSITION AND PHARMACEUTICAL USE THEREOF 长春金赛药业有限责任公司 2024-05-23 WO disclosed