SCHEMBL30952437

SCHEMBL30952437

COc1cccc(C2=CCCN(C(=O)OC(C)(C)C)C2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGAT2 Q10469 1/20 0.44
DGAT2 Q96PD7 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ABL1 P00519 1/20 0.44
EGFR P00533 1/20 0.44
SRC P12931 1/20 0.44
ABL2 P42684 1/20 0.44
USP30 Q70CQ3 2/20 0.44
MKNK1 Q9BUB5 1/20 0.42
ALDH1A1 P00352 1/20 0.41
ESR2 Q92731 1/20 0.41
TGFBR1 P36897 1/20 0.41
STS P08842 1/20 0.41
MAPK1 P28482 1/20 0.40
NR1H2 P55055 1/20 0.40
PDK4 Q16654 1/20 0.40
EPHX2 P34913 1/20 0.40
P2RX3 P56373 1/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21361618 1.00 MGAT2 (0.44) MGAT2DGAT2MEN1KMT2AABL1
SCHEMBL21425203 0.89 MAPK1 (0.41) MGAT2DGAT2USP30ESR2MAPK1
SCHEMBL29941117 0.88 PDK4 (0.47) MGAT2DGAT2MEN1KMT2AABL1
SCHEMBL21767871 0.88 PDK4 (0.47) MGAT2DGAT2MEN1KMT2AABL1
SCHEMBL15649776 0.88 ALDH1A1 (0.43) ALDH1A1ESR2STSMAPK1NR1H2
SCHEMBL22945388 0.86 USP30 (0.48) USP30ESR2MAPK1NR1H2PDK4
SCHEMBL31334489 0.85 USP30 (0.45) DGAT2MEN1KMT2AUSP30ESR2
SCHEMBL11195135 0.85 ALDH1A1 (0.48) MEN1KMT2AALDH1A1MAPK1KDM4E
SCHEMBL28516672 0.84 NCOA1 (0.44) MEN1KMT2AALDH1A1KDM4EMAPT
SCHEMBL6352947 0.84 MAPK1 (0.49) USP30ESR2MAPK1NR1H2PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112262129-B Triazacyclododecanesulfonamide (\"TCD\") based protein secretion inhibitors 科智生命科学公司 2024-05-14 CN disclosed