SCHEMBL30955022

SCHEMBL30955022

Cc1cnc(Cl)c(-c2c(F)cc(F)cc2F)c1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.34
CCR5 P51681 1/20 0.34
CCR8 P51685 1/20 0.34
GABRA1 P14867 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA5 P31644 1/20 0.31
GABRA3 P34903 1/20 0.31
GABRA2 P47869 1/20 0.31
KMT2A Q03164 1/20 0.31
RAPGEF4 Q8WZA2 2/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30954963 0.84 CCR1 (0.37) CCR1CCR5CCR8KMT2A
SCHEMBL30954959 0.79 NOS3 (0.47) CCR1CCR5CCR8GABRA1GABRG2
SCHEMBL30954977 0.75 BTK (0.33) CCR1CCR5CCR8
SCHEMBL17892 0.74
SCHEMBL29196121 0.73 HTR5A (0.34)
SCHEMBL30824457 0.73 HTR5A (0.34)
SCHEMBL30955012 0.69 ALOX5AP (0.36) NPC1RAB9A
SCHEMBL22326614 0.66 CCR1 (0.54) CCR1CCR5CCR8KMT2ARAPGEF4
SCHEMBL29184390 0.66 KMT2A (0.36) KMT2ARAPGEF4RAB9A
SCHEMBL15908809 0.66 CCR1 (0.39) CCR1CCR5CCR8NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4626546-A1 HETEROCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2025-10-08 EP disclosed
WO-2024116086-A1 HETEROCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2024-06-06 WO disclosed