SCHEMBL30957563

SCHEMBL30957563

COc1ccc2c(c1)c(-c1nc(Cl)ncc1F)cn2C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.49
GSK3B P49841 3/20 0.47
LCK P06239 2/20 0.47
IGF1R P08069 2/20 0.47
GSK3A P49840 2/20 0.47
CDK7 P50613 2/20 0.47
LRRK2 Q5S007 2/20 0.47
AURKB Q96GD4 2/20 0.47
AURKA O14965 1/20 0.47
PAK4 O96013 1/20 0.47
ABL1 P00519 1/20 0.47
NTRK1 P04629 1/20 0.47
FYN P06241 1/20 0.47
CSF1R P07333 1/20 0.47
RET P07949 1/20 0.47
MET P08581 1/20 0.47
PDGFRB P09619 1/20 0.47
PIM1 P11309 1/20 0.47
FGFR1 P11362 1/20 0.47
PRKACA P17612 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24900439 1.00 PDK1 (0.49) PDK1GSK3BLCKIGF1RGSK3A
SCHEMBL30957637 0.85 PDK1 (0.50) PDK1GSK3BLCKIGF1RGSK3A
SCHEMBL17490480 0.85 PDK1 (0.50) PDK1GSK3BLCKIGF1RGSK3A
SCHEMBL30221565 0.85 PDK1 (0.47) PDK1GSK3BLCKIGF1RGSK3A
SCHEMBL24900656 0.85 PDK1 (0.47) PDK1GSK3BLCKIGF1RGSK3A
SCHEMBL30957512 0.84 PDK1 (0.39) PDK1GSK3BLCKIGF1RGSK3A
SCHEMBL24900722 0.84 PDK1 (0.39) PDK1GSK3BLCKIGF1RGSK3A
SCHEMBL17490484 0.81 SMN1; SMN2 (0.38) PDK1GSK3BLCKIGF1RGSK3A
SCHEMBL30957490 0.81 SMN1; SMN2 (0.38) PDK1GSK3BLCKIGF1RGSK3A
SCHEMBL518274 0.80 CDK5 (0.51) PDK1CDK5CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118159533-A Heterocyclic compounds and their use 艾森医药有限公司 2024-06-07 CN disclosed