SCHEMBL30965261

SCHEMBL30965261

CCCCCCOc1cc2c(cc1[N+](=O)[O-])C(=O)N(CC(=O)O)C2=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.46
THRB P10828 1/20 0.46
PLA2G4B P0C869 1/20 0.45
ESR1 P03372 1/20 0.43
LPAR3 Q9UBY5 2/20 0.43
LMNA P02545 3/20 0.42
ALDH1A1 P00352 1/20 0.42
AGTR1 P30556 1/20 0.42
CYSLTR2 Q9NS75 1/20 0.41
CYSLTR1 Q9Y271 1/20 0.41
MAPT P10636 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
RAB9A P51151 1/20 0.40
PLA2G2A P14555 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30965272 0.89 THRA (0.47) THRATHRBPLA2G4BESR1LMNA
SCHEMBL30965271 0.88 THRA (0.46) THRATHRBPLA2G4BESR1LMNA
SCHEMBL30965267 0.84 LPAR3 (0.45) LPAR3LMNAALDH1A1AGTR1MAPT
SCHEMBL30965219 0.81 TDP1 (0.43) THRATHRBLPAR3LMNAALDH1A1
SCHEMBL30965265 0.81 HPGD (0.47) LPAR3LMNAALDH1A1AGTR1CYSLTR2
SCHEMBL30965202 0.77 TDP1 (0.40) THRATHRBLPAR3ALDH1A1PLA2G2A
SCHEMBL9322138 0.76 THRA (0.54) THRATHRBPLA2G4BESR1LMNA
SCHEMBL30965244 0.76 CYP19A1 (0.47) LPAR3ALDH1A1RAB9APLA2G2ATDP1
SCHEMBL30965165 0.73 ALDH1A1 (0.47) LMNAALDH1A1AGTR1CYSLTR2CYSLTR1
SCHEMBL30965155 0.72 ALDH1A1 (0.47) LMNAALDH1A1AGTR1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118125964-A Isoindoline-1, 3-diketone mPGES-1 inhibitor and application thereof 长江大学 2024-06-04 CN disclosed