SCHEMBL30968100

SCHEMBL30968100

Cc1nc([C@@H]2C[C@H]2c2ccc(C(=O)N(C)C3C[C@H]4CC[C@@H](C3)N4)cc2Cl)c2ccccc2n1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTAFR P25105 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
HRH3 Q9Y5N1 5/20 0.34
ADRA2A P08913 1/20 0.34
MCHR1 Q99705 1/20 0.34
GPR142 Q7Z601 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 1/20 0.33
PARP1 P09874 1/20 0.33
CHRM4 P08173 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30968132 1.00 PTAFR (0.35) PTAFROPRM1OPRD1HRH3ADRA2A
SCHEMBL30968042 1.00 PTAFR (0.35) PTAFROPRM1OPRD1HRH3ADRA2A
SCHEMBL30967987 0.88 PTAFR (0.36) PTAFROPRM1OPRD1HRH3ADRA2A
SCHEMBL30968105 0.88 POLB (0.32) OPRM1OPRD1GPR142
SCHEMBL31065783 0.85 PLD3 (0.32) GPR142
SCHEMBL31065780 0.85 PLD3 (0.32) GPR142
SCHEMBL31065775 0.85 PLD3 (0.32) GPR142
SCHEMBL30968089 0.84 PARP1 (0.33) PTAFRHRH3ADRA2AMCHR1GPR142
SCHEMBL30968015 0.84 PARP1 (0.33) PTAFRHRH3ADRA2AMCHR1GPR142
SCHEMBL30968069 0.81 MAPK1 (0.38) ADRA2AMCHR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024131942-A1 CYCLOPROPANE TLR7 AND TLR8 INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF 上海深势唯思科技有限责任公司 2024-06-27 WO disclosed
CN-118239959-A Cyclopropane TLR7 and 8 inhibitor and preparation method and application thereof 上海深势唯思科技有限责任公司 2024-06-25 CN disclosed