SCHEMBL30970478

SCHEMBL30970478

C=C(F)C(=O)Nc1cccc2c1CN(C(=O)c1c(O)cc(O)cc1OCc1ccccc1)C2

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRAP1 Q12931 6/20 0.36
HSP90B1 P14625 4/20 0.36
BRD4 O60885 1/20 0.35
NAMPT P43490 1/20 0.34
HSP90AA1 P07900 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
SPR P35270 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PPIA P62937 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
TSHR P16473 1/20 0.34
HSP90AB1 P08238 1/20 0.33
SLC6A9 P48067 1/20 0.33
SLC5A1 P13866 1/20 0.33
SLC5A2 P31639 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25248972 1.00 TRAP1 (0.36) TRAP1HSP90B1BRD4NAMPTHSP90AA1
SCHEMBL25253974 0.88 TGM2 (0.39) TRAP1HSP90B1BRD4NAMPTSLC5A1
SCHEMBL30970470 0.88 TGM2 (0.39) TRAP1HSP90B1BRD4NAMPTSLC5A1
SCHEMBL29168554 0.88 BRD4 (0.49) TRAP1HSP90B1BRD4
SCHEMBL30970496 0.86 GLRA1 (0.35) TRAP1HSP90B1HSP90AA1SPRALDH1A1
SCHEMBL25211585 0.86 GLRA1 (0.35) TRAP1HSP90B1HSP90AA1SPRALDH1A1
SCHEMBL24913934 0.86 TRAP1 (0.41) TRAP1HSP90B1BRD4HSP90AA1L3MBTL1
SCHEMBL30789151 0.86 TRAP1 (0.41) TRAP1HSP90B1BRD4HSP90AA1L3MBTL1
SCHEMBL24913881 0.81 TRAP1 (0.51) TRAP1HSP90B1HSP90AA1L3MBTL1SPR
SCHEMBL30156809 0.81 TRAP1 (0.51) TRAP1HSP90B1HSP90AA1L3MBTL1SPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118317949-A Isoindolines as PMS2 inhibitors 奈奥芬莱有限公司 2024-07-09 CN claimed
CN-118317949-A Isoindolines as PMS2 inhibitors 奈奥芬莱有限公司 2024-07-09 CN disclosed