SCHEMBL30979817

SCHEMBL30979817

Cc1cn(-c2ccc(C(F)(F)F)nc2)nn1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.43
TRPV4 Q9HBA0 1/20 0.41
RXRA P19793 6/20 0.40
GRIN1 Q05586 6/20 0.40
GRIN2B Q13224 6/20 0.40
PTGS2 P35354 4/20 0.39
KCNH2 Q12809 1/20 0.39
AR P10275 3/20 0.37
DHFR P00374 1/20 0.37
PTGS1 P23219 1/20 0.36
LRRK2 Q5S007 1/20 0.36
MAT2A P31153 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23999583 0.80 DDX3X (0.41) NOTUMRXRAGRIN1GRIN2BLRRK2
SCHEMBL21263902 0.77 NOTUM (0.59) NOTUMRXRAGRIN1GRIN2BPTGS2
SCHEMBL15935031 0.76 HTT (0.46) TRPV4PTGS2DHFRPTGS1MAT2A
SCHEMBL18086468 0.76 KDM4E (0.42) TRPV4PTGS2DHFRPTGS1
SCHEMBL29640824 0.76 MAPT (0.44) NOTUMRXRAGRIN1GRIN2BLRRK2
SCHEMBL21275488 0.76 MAPT (0.44) NOTUMRXRAGRIN1GRIN2BLRRK2
SCHEMBL26847601 0.75 TRPV4 (0.41) TRPV4PTGS2DHFRPTGS1MAT2A
SCHEMBL25043775 0.75 GRIN1 (0.38) NOTUMRXRAGRIN1GRIN2BKCNH2
SCHEMBL30343244 0.75 GRIN1 (0.38) NOTUMRXRAGRIN1GRIN2BKCNH2
SCHEMBL25408961 0.73 DHFR (0.41) TRPV4PTGS2KCNH2DHFRPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118284606-A Bicyclic amine derivatives as GABAA α5 receptor modulators 吉瑞工厂 2024-07-02 CN disclosed