SCHEMBL30982104

SCHEMBL30982104

CN(C)C(=O)CNCC(c1ccccc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 2/20 0.48
GRIN1 Q05586 2/20 0.44
GRIN2A Q12879 2/20 0.44
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
CYP2D6 P10635 2/20 0.43
KMT2A Q03164 2/20 0.42
HTR2A P28223 1/20 0.41
HRH1 P35367 1/20 0.41
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
MEN1 O00255 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
APAF1 O14727 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
KCNH2 Q12809 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7394409 0.87 TAAR1 (0.47) CACNA1BALDH1A1KDM4EL3MBTL1CYP2D6
SCHEMBL7394405 0.87 TAAR1 (0.47) CACNA1BALDH1A1KDM4EL3MBTL1CYP2D6
Hydrochloric Acid SCHEMBL4228085 0.84 PPIB (0.45) GRIN1GRIN2AALDH1A1KDM4EL3MBTL1
Hydrochloric Acid SCHEMBL4236478 0.80 NPSR1 (0.47) CACNA1BGRIN1GRIN2AALDH1A1KDM4E
SCHEMBL181573 0.80 GRIN1 (0.52) GRIN1GRIN2AKDM4EL3MBTL1CYP2D6
Hydrochloric Acid SCHEMBL4226515 0.79 ALDH1A1 (0.55) GRIN1GRIN2AALDH1A1KDM4EL3MBTL1
SCHEMBL30982190 0.78 KMT2A (0.53) CACNA1BKDM4EKMT2AMEN1SLC6A3
SCHEMBL31477970 0.77 KMT2A (0.52) GRIN1GRIN2AALDH1A1L3MBTL1KMT2A
SCHEMBL7310631 0.77 BCAT2 (0.49) GRIN1GRIN2AALDH1A1KDM4EL3MBTL1
SCHEMBL7391860 0.76 APAF1 (0.56) ALDH1A1KDM4ECYP2D6KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024153595-A1 CHROMANE DERIVATIVES AS EGFR SELECTIVE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2024-07-25 WO disclosed