SCHEMBL30987404

SCHEMBL30987404

COc1ccc(S(=O)(=O)Nc2ccc(NC(=O)c3ccccc3C)c3ccccc23)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 12/20 0.68
NFE2L2 Q16236 6/20 0.68
SQSTM1 Q13501 1/20 0.68
LMNA P02545 4/20 0.63
ALDH1A1 P00352 3/20 0.63
SMN1; SMN2 Q16637 3/20 0.63
MAPT P10636 2/20 0.63
TP53 P04637 2/20 0.63
HPGD P15428 2/20 0.63
L3MBTL1 Q9Y468 2/20 0.63
MITF O75030 1/20 0.63
GAA P10253 1/20 0.63
THRB P10828 1/20 0.63
ALOX15 P16050 1/20 0.63
CASP1 P29466 1/20 0.63
GFER P55789 1/20 0.63
HKDC1 Q2TB90 1/20 0.63
HSD17B10 Q99714 1/20 0.63
NPC1 O15118 1/20 0.56
RAB9A P51151 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8627655 0.90 KEAP1 (0.67) KEAP1NFE2L2SQSTM1LMNAALDH1A1
SCHEMBL27295108 0.88 FLT1 (0.54) KEAP1NFE2L2SQSTM1LMNAALDH1A1
SCHEMBL30987388 0.88 FLT1 (0.54) KEAP1NFE2L2SQSTM1LMNAALDH1A1
SCHEMBL30987406 0.84 CCR8 (0.75) LMNAALDH1A1SMN1; SMN2MAPTHSD17B10
SCHEMBL1340327 0.84 CCR8 (0.75) LMNAALDH1A1SMN1; SMN2MAPTHSD17B10
SCHEMBL26089402 0.83 KEAP1 (1.00) KEAP1NFE2L2SQSTM1LMNAALDH1A1
SCHEMBL8627716 0.81 TUBB4A (0.59) KEAP1LMNAALDH1A1SMN1; SMN2MAPT
SCHEMBL29892528 0.80 KEAP1 (0.77) KEAP1NFE2L2SQSTM1LMNAALDH1A1
SCHEMBL28841732 0.78 KEAP1 (0.70) KEAP1NFE2L2SQSTM1LMNAALDH1A1
SCHEMBL21511039 0.78 GAA (1.00) KEAP1NFE2L2SQSTM1LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024133292-A1 NOVEL CCR8 ANTAGONISTS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2024-06-27 WO disclosed