SCHEMBL30998202

SCHEMBL30998202

C[Si](C)(C)C#Cc1ccc(COS(C)(=O)=O)nc1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 6/20 0.35
GABRG2 P18507 6/20 0.35
GABRB3 P28472 6/20 0.35
GABRA5 P31644 6/20 0.35
GABRA3 P34903 6/20 0.35
GABRA2 P47869 6/20 0.35
GABRA4 P48169 4/20 0.35
GABRA6 Q16445 4/20 0.35
GRM5 P41594 1/20 0.34
FFAR1 O14842 1/20 0.34
ACACB O00763 1/20 0.34
LOX P28300 1/20 0.33
GABRB2 P47870 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18443081 0.81 RORC (0.39) GABRA5
SCHEMBL29241068 0.79 CA2 (0.39) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL30998309 0.77 FFAR1 (0.34) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL30998279 0.77 FFAR1 (0.34) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL29022647 0.76 GABRA1 (0.41) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL5096641 0.75 FFAR1 (0.37) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL3001118 0.73 FFAR1 (0.40) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL12661548 0.73 SYK (0.39) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL15986833 0.72 CYP1A2 (0.32)
SCHEMBL506719 0.72 HTR2A (0.39) GABRA5ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024153173-A1 AROMATIC ACETYLENE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 浙江海正药业股份有限公司 2024-07-25 WO disclosed