SCHEMBL31006887

SCHEMBL31006887

Cc1nc(=O)c2c([nH]1)CN(C(=O)OC(C)(C)C)CC2

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.44
TNKS2 Q9H2K2 1/20 0.44
PARP2 Q9UGN5 1/20 0.44
ADORA1 P30542 2/20 0.43
ESR2 Q92731 1/20 0.41
NR1H2 P55055 1/20 0.40
F12 P00748 3/20 0.39
MAPT P10636 2/20 0.39
TRPV1 Q8NER1 2/20 0.38
SPR P35270 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPK1 P28482 1/20 0.38
GRM5 P41594 1/20 0.36
P2RX3 P56373 1/20 0.36
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
FABP4 P15090 1/20 0.36
FABP5 Q01469 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13250475 0.80 PARP1 (0.51) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL31138807 0.78 ADORA1 (0.45) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL2456754 0.78 SPR (0.46) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL30474108 0.78 ESR2 (0.46) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL2191982 0.76 DDB1 (0.38) PARP1TNKS2PARP2NR1H2MAPT
SCHEMBL17229883 0.75 ADORA1 (0.45) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL29689663 0.75 ADORA1 (0.47) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL2270578 0.73 PARP1 (0.57) PARP1TNKS2PARP2TRPV1MAPK1
SCHEMBL123032 0.73 ESR2 (0.54) PARP1TNKS2PARP2ADORA1ESR2
SCHEMBL1967387 0.73 ADORA1 (0.45) PARP1TNKS2PARP2ADORA1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118480029-A 2-Aminopyrimidine compound or salt thereof, and preparation method and application thereof 励缔(杭州)医药科技有限公司 2024-08-13 CN disclosed