SCHEMBL31008705

SCHEMBL31008705

COc1ccc(Cn2c(=O)[nH]c3cc(-c4ccc(F)cc4)cnc32)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 8/20 0.59
GRIN2B Q13224 8/20 0.59
KDM4E B2RXH2 2/20 0.51
MTOR P42345 1/20 0.51
ALDH1A1 P00352 6/20 0.50
CYP1A2 P05177 3/20 0.50
CNR2 P34972 2/20 0.50
CASP1 P29466 2/20 0.50
HSD17B10 Q99714 2/20 0.50
USP2 O75604 2/20 0.50
CYP3A4 P08684 2/20 0.50
CNR1 P21554 1/20 0.50
MEN1 O00255 1/20 0.49
MAPT P10636 1/20 0.49
KMT2A Q03164 1/20 0.49
HPGD P15428 2/20 0.48
NPSR1 Q6W5P4 1/20 0.48
HIF1A Q16665 2/20 0.48
CASP7 P55210 1/20 0.48
CYP2C9 P11712 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21117369 0.84 PDE4B (0.61) GRIN1GRIN2BHSD17B10
SCHEMBL20129909 0.81 PDE1B (0.56) GRIN1GRIN2BKDM4EMTORALDH1A1
SCHEMBL29636174 0.81 PDE1B (0.56) GRIN1GRIN2BKDM4EMTORALDH1A1
SCHEMBL17242598 0.78 KDM4E (0.70) KDM4EALDH1A1CASP1HSD17B10USP2
SCHEMBL34462136 0.76 ALDH1A1 (0.55) GRIN1GRIN2BKDM4EMTORALDH1A1
SCHEMBL29722691 0.75 KDM4E (0.56) KDM4EMTORALDH1A1MEN1MAPT
SCHEMBL21117546 0.75 PDE4B (0.62) GRIN1GRIN2BHSD17B10
SCHEMBL20134563 0.74 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL18556093 0.73 GRIN1 (0.58) GRIN1GRIN2BKDM4EMTORALDH1A1
SCHEMBL29691179 0.73 KDM4E (0.54) GRIN1GRIN2BKDM4EMTORALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114989164-B Substituted 1H-imidazo [4,5-b ] pyridin-2 (3H) -ones and uses thereof 詹森药业有限公司 2024-08-13 CN disclosed