SCHEMBL31016830

SCHEMBL31016830

O=C1c2ccccc2C(=O)N1CC=C(F)F

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.51
CA12 O43570 1/20 0.48
CA9 Q16790 1/20 0.48
ALDH1A1 P00352 2/20 0.46
GLS O94925 1/20 0.44
NPSR1 Q6W5P4 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.42
MAPK1 P28482 1/20 0.42
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8533004 0.81 GLS (0.50) CA12CA9GLS
SCHEMBL29486825 0.81 CASP3 (0.45) CASP3CA12CA9ALDH1A1GLS
SCHEMBL28720232 0.81 CASP3 (0.45) CASP3CA12CA9ALDH1A1GLS
SCHEMBL22918274 0.81 CASP3 (0.45) CASP3CA12CA9ALDH1A1GLS
SCHEMBL4017572 0.81 ALDH1A1 (0.55) CASP3CA12CA9ALDH1A1GLS
SCHEMBL16623099 0.78 ALDH1A1 (0.51) CASP3CA12CA9ALDH1A1GLS
SCHEMBL11109119 0.77 CASP3 (0.42) CASP3CA12CA9ALDH1A1KDM4E
SCHEMBL4476083 0.77 CASP3 (0.60) CASP3CA12CA9ALDH1A1GLS
SCHEMBL4468251 0.77 CASP3 (0.60) CASP3CA12CA9ALDH1A1GLS
SCHEMBL8950475 0.77 CASP3 (0.60) CASP3CA12CA9ALDH1A1GLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024217500-A1 ISOQUINOLINE COMPOUND, AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND USE THEREOF 上海赛默罗生物科技有限公司 2024-10-24 WO disclosed
CN-118359538-A Isoquinoline compound, preparation method, pharmaceutical composition and application thereof 上海赛默罗生物科技有限公司 2024-07-19 CN disclosed