SCHEMBL31035879

SCHEMBL31035879

C#CCN(CC(=O)O)C(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 1/20 0.42
CES2 O00748 2/20 0.42
CES1 P23141 2/20 0.42
POLQ O75417 1/20 0.42
SRD5A2 P31213 2/20 0.41
PTPN1 P18031 2/20 0.41
GSK3B P49841 1/20 0.41
LIMK1 P53667 1/20 0.40
LIMK2 P53671 1/20 0.40
HSD11B1 P28845 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
MLYCD O95822 2/20 0.39
NR4A1 P22736 1/20 0.38
NR4A2 P43354 1/20 0.38
NR4A3 Q92570 1/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31036190 0.86 MLYCD (0.45) CES2CES1POLQSRD5A2PTPN1
SCHEMBL31035930 0.86 NR1H4 (0.46) SRD5A2LIMK1LIMK2
SCHEMBL31035978 0.78 MEN1 (0.54) MEN1KMT2AMLYCD
SCHEMBL31035948 0.76 MAPT (0.49) SRD5A2MEN1KMT2A
SCHEMBL31035945 0.75 MLYCD (0.52) CES2CES1SRD5A2PTPN1MEN1
SCHEMBL31035814 0.74 PYCR1 (0.56) PYCR1POLQSRD5A2PTPN1GSK3B
SCHEMBL24457331 0.74 CES2 (0.39) CES2CES1SRD5A2PTPN1GSK3B
SCHEMBL7281175 0.72 MLYCD (0.69) CES2CES1PTPN1GSK3BMEN1
SCHEMBL31035984 0.71 NR1H4 (0.46) SRD5A2MLYCD
SCHEMBL8484820 0.71 LIMK1 (0.52) LIMK1LIMK2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118459520-A Spiramycin acylated derivative, preparation method, application and pharmaceutical composition 赣江中药创新中心 2024-08-09 CN disclosed