SCHEMBL31038488

SCHEMBL31038488

Nc1cccc2cccc(Br)c12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.45
RPS6KA3 P51812 1/20 0.45
MELK Q14680 1/20 0.45
STK24 Q9Y6E0 1/20 0.45
BACE1 P56817 2/20 0.43
CYP3A4 P08684 6/20 0.42
ALDH1A1 P00352 6/20 0.42
TSHR P16473 5/20 0.42
HSD17B10 Q99714 5/20 0.42
HPGD P15428 3/20 0.42
KEAP1 Q14145 1/20 0.42
CYP1A2 P05177 2/20 0.41
CYP1A1 P04798 1/20 0.41
CYP1B1 Q16678 1/20 0.41
AXL P30530 1/20 0.41
TYMS P04818 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MEN1 O00255 2/20 0.37
GAA P10253 2/20 0.37
KMT2A Q03164 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4087754 1.00 JAK2 (0.45) JAK2RPS6KA3MELKSTK24BACE1
SCHEMBL29374267 0.81 ALDH1A1 (0.53) BACE1CYP3A4ALDH1A1TSHRHSD17B10
SCHEMBL29349435 0.81 JAK2 (0.54) JAK2RPS6KA3MELKSTK24CYP3A4
SCHEMBL1187339 0.81 ALDH1A1 (0.53) BACE1CYP3A4ALDH1A1TSHRHSD17B10
SCHEMBL65699 0.81 JAK2 (0.54) JAK2RPS6KA3MELKSTK24CYP3A4
SCHEMBL8878160 0.79 CYP3A4 (0.42) JAK2RPS6KA3MELKSTK24BACE1
SCHEMBL14742902 0.78 ALDH1A1 (0.59) JAK2RPS6KA3MELKSTK24CYP3A4
Hydrochloric Acid SCHEMBL11277860 0.78 JAK2 (0.52) JAK2RPS6KA3MELKSTK24CYP3A4
Ammonia Solution, Strong SCHEMBL2638226 0.78 JAK2 (0.52) JAK2RPS6KA3MELKSTK24CYP3A4
SCHEMBL9627127 0.78 JAK2 (0.52) JAK2RPS6KA3MELKSTK24CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118451068-A Tri-fused ring derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-08-06 CN disclosed