SCHEMBL31048007

SCHEMBL31048007

COC(=O)c1ccc(NC2CN(C(=O)OC(C)(C)C)C2)c(C)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.44
EHMT2 Q96KQ7 1/20 0.43
PIM1 P11309 1/20 0.41
PIM2 Q9P1W9 1/20 0.41
ALDH1A1 P00352 2/20 0.41
GPR119 Q8TDV5 1/20 0.41
USP30 Q70CQ3 5/20 0.39
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SSTR4 P31391 1/20 0.38
PDE4B Q07343 1/20 0.38
EGFR P00533 1/20 0.37
ERBB2 P04626 1/20 0.37
ERBB3 P21860 1/20 0.37
ERBB4 Q15303 1/20 0.37
BRD4 O60885 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31048018 0.88 PIM1 (0.41) EHMT2PIM1PIM2ALDH1A1USP30
SCHEMBL31048004 0.88 PIM1 (0.41) EHMT2PIM1PIM2ALDH1A1USP30
SCHEMBL31178709 0.82 PDE4B (0.43) NR1H2GPR119SSTR4PDE4B
SCHEMBL16834214 0.81 NR1H2 (0.45) NR1H2EHMT2PIM1PIM2ALDH1A1
SCHEMBL30849213 0.80 ALDH1A1 (0.47) NR1H2ALDH1A1GPR119USP30NPC1
SCHEMBL25191571 0.78 GPR119 (0.50) NR1H2EHMT2ALDH1A1GPR119USP30
SCHEMBL30234604 0.78 GPR119 (0.50) NR1H2EHMT2ALDH1A1GPR119USP30
SCHEMBL31358059 0.78 USP30 (0.45) NR1H2PIM1PIM2ALDH1A1GPR119
SCHEMBL24157379 0.78 NR1H2 (0.49) NR1H2ALDH1A1GPR119MAPT
SCHEMBL30297083 0.78 NR1H2 (0.49) NR1H2ALDH1A1GPR119MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024178125-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF 1CBIO, INC. (US) 2024-08-29 WO disclosed