SCHEMBL31064153

SCHEMBL31064153

CSc1nc(NC2CCC(C(=O)OC3CCN(C(=O)OCc4ccccc4)C3)CC2)n2ncc(C(C)C)c2n1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 7/20 0.41
CDK7 P50613 6/20 0.41
CDK4 P11802 1/20 0.41
CDK2 P24941 7/20 0.40
PIK3CD O00329 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
CCNH P51946 5/20 0.37
MNAT1 P51948 5/20 0.37
CYP2C19 P33261 1/20 0.37
HTT P42858 1/20 0.37
ENPP2 Q13822 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31064534 0.89 CDK9 (0.41) CDK9CDK7CDK4CDK2PIK3CD
SCHEMBL31064105 0.87 CDK2 (0.51) CDK9CDK7CDK4CDK2CCNH
SCHEMBL31064107 0.86 CDK9 (0.42) CDK9CDK7CDK4CDK2PIK3CD
SCHEMBL31064465 0.76 CDK2 (0.41) CDK9CDK7CDK4CDK2
SCHEMBL23547341 0.74 ALDH1A1 (0.49) CDK9CDK7CDK4CDK2NPC1
SCHEMBL31064296 0.69 CDK7 (0.50) CDK9CDK7CDK4CDK2CCNH
SCHEMBL31064118 0.69 CDK4 (0.51) CDK9CDK7CDK4PIK3CDNPC1
SCHEMBL23547346 0.69 CDK9 (0.51) CDK9CDK7CDK4CDK2NPC1
SCHEMBL23529883 0.68 CDK9 (0.54) CDK9CDK7CDK4CDK2PIK3CD
SCHEMBL31064099 0.67 CDK9 (0.49) CDK9CDK7CDK4CDK2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024175024-A1 NEW FUSED HETEROCYCLIC COMPOUND AS CDKS INHIBITOR AND USE THEREOF 杭州德睿智药科技有限公司 2024-08-29 WO disclosed