SCHEMBL31064465

SCHEMBL31064465

CSc1nc(NC2CCC(C(=O)O)CC2)n2ncc(C(C)C)c2n1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 17/20 0.41
CDK9 P50750 17/20 0.41
CDK4 P11802 2/20 0.41
CDK7 P50613 2/20 0.41
SRC P12931 1/20 0.39
PDE7A Q13946 1/20 0.38
ADORA1 P30542 1/20 0.35
DYRK3 O43781 1/20 0.35
CCNT1 O60563 1/20 0.35
CCNA2 P20248 1/20 0.35
CLK1 P49759 1/20 0.35
CLK2 P49760 1/20 0.35
CLK3 P49761 1/20 0.35
CDK5 Q00535 1/20 0.35
DYRK1A Q13627 1/20 0.35
CDK5R1 Q15078 1/20 0.35
DYRK2 Q92630 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
DYRK1B Q9Y463 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23547341 0.79 ALDH1A1 (0.49) CDK2CDK9CDK4CDK7CCNA2
SCHEMBL31064107 0.77 CDK9 (0.42) CDK2CDK9CDK4CDK7
SCHEMBL31064134 0.76 KAT2B (0.42) CDK2CDK9CDK4CDK7
SCHEMBL31064153 0.76 CDK9 (0.41) CDK2CDK9CDK4CDK7
SCHEMBL31064144 0.75 CDK2 (0.43) CDK2CDK9CDK4CDK7CCNT1
SCHEMBL16659551 0.75 CDK2 (0.36) CDK2CDK9CDK7SRCCCNT1
SCHEMBL1486116 0.72 CSNK2B (0.50) SRCPDE7AADORA1
SCHEMBL19912801 0.72 CDK2 (0.41) CDK2CDK9CDK4CDK7ADORA1
SCHEMBL23547517 0.72 CDK9 (0.45) CDK2CDK9CDK4CDK7
SCHEMBL15241430 0.72 CDK2 (0.40) CDK2CDK9CDK4CDK7SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024175024-A1 NEW FUSED HETEROCYCLIC COMPOUND AS CDKS INHIBITOR AND USE THEREOF 杭州德睿智药科技有限公司 2024-08-29 WO disclosed