SCHEMBL31069265

SCHEMBL31069265

CCc1cccc(-c2c(C(=O)O)nn3c2COCC3)n1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 6/20 0.37
THRB P10828 2/20 0.37
MAPK14 Q16539 1/20 0.37
AOC3 Q16853 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
KCNK3 O14649 6/20 0.33
ACVR1 Q04771 5/20 0.33
GRM5 P41594 2/20 0.33
GRM1 Q13255 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23645337 1.00 TGFBR1 (0.37) TGFBR1THRBMAPK14AOC3CCNE1
SCHEMBL23652810 0.85 TGFBR1 (0.39) TGFBR1THRBMAPK14ACVR1GRM5
SCHEMBL20213765 0.76 PTPN1 (0.40) ACVR1
SCHEMBL21315407 0.73 KCNK3 (0.33) KCNK3
SCHEMBL23645307 0.66 POLB (0.31)
SCHEMBL23652637 0.66
SCHEMBL24581298 0.63 ECE1 (0.54)
SCHEMBL12359155 0.62 IRAK4 (0.49)
SCHEMBL22767997 0.61 KMT2A (0.43)
SCHEMBL6200651 0.61 RAB9A (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112689636-B Novel heteroatom aromatic amide derivative and pharmaceutical agent containing same 科研制药株式会社 2024-08-20 CN disclosed