SCHEMBL31069446

SCHEMBL31069446

Cn1c(=O)n(Cc2cc3cc(CNC(=O)OC(C)(C)C)ccc3n2CCCS(C)(=O)=O)c2cc(F)ccc21

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GNRHR P30968 1/20 0.38
GRM2 Q14416 1/20 0.36
KDM4E B2RXH2 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
PLK1 P53350 4/20 0.35
BRD4 O60885 1/20 0.35
BRD9 Q9H8M2 1/20 0.34
BAZ2B Q9UIF8 1/20 0.34
BAZ2A Q9UIF9 1/20 0.34
TP53 P04637 3/20 0.34
EPHX2 P34913 1/20 0.34
PPARG P37231 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
LMNA P02545 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31069447 0.89 GRM2 (0.37) GNRHRGRM2KDM4ECYP1A2CYP3A4
SCHEMBL31069392 0.82 PARG (0.36)
SCHEMBL31069450 0.78 PARG (0.34)
SCHEMBL31069497 0.75 GNRHR (0.47) GNRHRGRM2KDM4ECYP1A2CYP3A4
SCHEMBL31069293 0.73 PTGS2 (0.33) CYP3A4
SCHEMBL15552909 0.73 P2RX3 (0.38) CYP3A4PLK1
SCHEMBL31069401 0.71 PTGS2 (0.32)
SCHEMBL31069459 0.71 KDM4E (0.41) GRM2KDM4ECYP1A2CYP3A4CYP2C19
SCHEMBL6242216 0.71 GNRHR (0.43) GNRHRGRM2CYP3A4CYP2C19BRD4
SCHEMBL31069325 0.71 PARG (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024174953-A1 BENZIMIDAZOLE DERIVATIVE AND MEDICAL USE THEREOF 苏州隆博泰药业有限公司 2024-08-29 WO disclosed