SCHEMBL31070073

SCHEMBL31070073

COCCC(=O)c1c[nH]c2nccc(Br)c12

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PKM P14618 4/20 0.53
MAP2K1 Q02750 1/20 0.40
CCNT1 O60563 1/20 0.37
CDK9 P50750 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
MAP3K7 O43318 2/20 0.36
TAB1 Q15750 2/20 0.36
BTK Q06187 4/20 0.36
JAK2 O60674 4/20 0.35
JAK3 P52333 2/20 0.34
UTS2R Q9UKP6 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21678497 1.00 PKM (0.53) PKMMAP2K1CCNT1CDK9CDK5
SCHEMBL21678385 0.83 PKM (0.53) PKMMAP2K1CDK9CDK5MAP3K7
SCHEMBL31070084 0.83 PKM (0.53) PKMMAP2K1CDK9CDK5MAP3K7
SCHEMBL30365873 0.81 MAP2K1 (0.56) PKMMAP2K1JAK2JAK3ALDH1A1
SCHEMBL22553986 0.81 MAP2K1 (0.56) PKMMAP2K1JAK2JAK3ALDH1A1
SCHEMBL30134852 0.78 MAP3K7 (0.45) PKMMAP2K1CDK9CDK5MAP3K7
SCHEMBL28994444 0.76 PKM (0.45) PKMMAP2K1CDK9CDK5JAK2
SCHEMBL23610513 0.75 PRKCI (0.45) PKMMAP2K1CDK9CDK5ALDH1A1
SCHEMBL857339 0.74 PKM (0.42) PKMMAP2K1CDK9CDK5JAK3
SCHEMBL21705113 0.73 ROCK2 (0.53) BTKJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119080779-A Pyrrolopyrimidine ITK inhibitors 阿克拉瑞斯治疗股份有限公司 2024-12-06 CN disclosed
CN-112823005-B Pyrrolopyrimidine ITK inhibitors 阿克拉瑞斯治疗股份有限公司 2024-08-20 CN disclosed