SCHEMBL31089289

SCHEMBL31089289

O=c1cc(C(F)(F)F)c(CCN2CCCC2)c[nH]1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MPO P05164 3/20 0.46
HTR1D P28221 8/20 0.43
HTR1B P28222 8/20 0.43
HTR2A P28223 5/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
HTR1A P08908 1/20 0.39
PIK3R1 P27986 1/20 0.38
PIK3CA P42336 1/20 0.38
AR P10275 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23249136 0.97 HTR2A (0.43) MPOHTR1DHTR1BHTR2AHTR2C
SCHEMBL27296035 0.89 MPO (0.45) MPOHTR1DHTR1BHTR2AHTR1A
SCHEMBL31089345 0.88 PIK3R1 (0.49) PIK3R1PIK3CA
SCHEMBL30972910 0.87 HTR1D (0.36) MPOHTR1DHTR1BPIK3R1PIK3CA
SCHEMBL27294746 0.83 GRIN1 (0.35) MPOPIK3R1PIK3CAAR
SCHEMBL27297250 0.83 PIK3R1 (0.34) MPOPIK3R1PIK3CA
SCHEMBL29725876 0.79 GRIN1 (0.37) MPOHTR2AHTR1APIK3R1PIK3CA
SCHEMBL12649073 0.72 HRH3 (0.53)
SCHEMBL30972827 0.72 CACNA1H (0.38) HTR2AHTR2CPIK3R1PIK3CAAR
SCHEMBL21459566 0.72 HTR1A (0.42) MPOHTR1DHTR1BHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024175907-A1 MACROCYCLIC ALPHA4BETA7 INTEGRIN INHIBITORS C4X DISCOVERY LIMITED (GB) 2024-08-29 WO disclosed