SCHEMBL31089345

SCHEMBL31089345

O=c1cc(C(F)(F)F)c(CCN2CCOCC2)c[nH]1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3R1 P27986 1/20 0.49
PIK3CA P42336 1/20 0.49
WDR5 P61964 15/20 0.41
PDE3B Q13370 2/20 0.41
PDE3A Q14432 2/20 0.41
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23249136 0.88 HTR2A (0.43) PIK3R1PIK3CA
SCHEMBL31089289 0.88 MPO (0.46) PIK3R1PIK3CA
SCHEMBL30972910 0.83 HTR1D (0.36) PIK3R1PIK3CA
SCHEMBL27294746 0.80 GRIN1 (0.35) PIK3R1PIK3CAWDR5
SCHEMBL27297250 0.80 PIK3R1 (0.34) PIK3R1PIK3CAWDR5
SCHEMBL27296035 0.80 MPO (0.45) PIK3R1PIK3CA
SCHEMBL29725876 0.76 GRIN1 (0.37) PIK3R1PIK3CAWDR5
SCHEMBL13071153 0.75 HRH3 (0.54) PDE3BPDE3AKMT2A
SCHEMBL27816674 0.71 HTR1D (0.49)
SCHEMBL21459566 0.69 HTR1A (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024175907-A1 MACROCYCLIC ALPHA4BETA7 INTEGRIN INHIBITORS C4X DISCOVERY LIMITED (GB) 2024-08-29 WO disclosed