SCHEMBL3109201

SCHEMBL3109201

CSCCc1c(C(=O)NCc2cccc(F)c2)nnn1-c1ccc(C(=O)NCC(F)(F)F)cc1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 3/20 0.46
ROCK2 O75116 4/20 0.41
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
NAMPT P43490 1/20 0.39
MLYCD O95822 1/20 0.39
ROCK1 Q13464 1/20 0.38
MMP13 P45452 1/20 0.38
ABCB1 P08183 1/20 0.38
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3113720 0.91 CCR1 (0.43) CCR1ROCK2TP53MAPTNAMPT
SCHEMBL5249091 0.87 CCR1 (0.44) CCR1ROCK2TP53MAPTNAMPT
SCHEMBL5245586 0.84 CCR1 (0.46) CCR1ROCK2TP53MAPTNAMPT
SCHEMBL3108441 0.83 CCR1 (0.47) CCR1ROCK2TP53MAPTNAMPT
SCHEMBL5244366 0.82 CCR1 (0.45) CCR1ROCK2TP53MAPTNAMPT
SCHEMBL3120022 0.82 CCR1 (0.39) CCR1ROCK2TP53MAPTNAMPT
SCHEMBL3119917 0.81 L3MBTL1 (0.37) CCR1TP53
SCHEMBL3111239 0.81 HPGD (0.39) TP53THRB
SCHEMBL3115763 0.79 CYP2C9 (0.37) TP53MAPT
SCHEMBL5243725 0.78 CCR1 (0.45) CCR1TP53MAPTMLYCDABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7803822-B2 Triazole derivative and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-28 US disclosed
US-20090105253-A1 Triazole Derivative and Use Thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-23 US disclosed
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090105253-A1 Triazole Derivative and Use Thereof F2R, HRH4, F2RL3 CCR1 184/4885ROCK2 2794/4885TP53 2716/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.