SCHEMBL3120022

SCHEMBL3120022

O=C(NCCNC(=O)c1nnn(-c2ccc(C(=O)NCC(F)(F)F)cc2)c1CCCCCF)NCc1cccc(F)c1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.39
ABCB1 P08183 1/20 0.39
MLYCD O95822 4/20 0.36
ROCK2 O75116 2/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
GLS O94925 1/20 0.35
NAMPT P43490 2/20 0.35
GABRA5 P31644 1/20 0.35
MMP13 P45452 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5249091 0.95 CCR1 (0.44) CCR1ABCB1MLYCDROCK2TP53
SCHEMBL3108829 0.89 NPC1 (0.40) MAPTNAMPTPOLB
SCHEMBL3107690 0.85 FOLH1 (0.33) CCR1MLYCD
SCHEMBL3104271 0.85 CYP1A2 (0.38) CCR1MLYCD
SCHEMBL5245660 0.84 MLYCD (0.50) MLYCDTP53NAMPTPOLB
SCHEMBL3112810 0.84 MLYCD (0.36) CCR1MLYCDMAPT
SCHEMBL3112218 0.83 RAB9A (0.36) MLYCD
SCHEMBL5246279 0.83 RAB9A (0.40) CCR1MLYCDMAPT
SCHEMBL3106801 0.83 HDAC4 (0.35) MLYCD
SCHEMBL5245108 0.83 NPC1 (0.37) MLYCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7803822-B2 Triazole derivative and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-28 US disclosed
US-20090105253-A1 Triazole Derivative and Use Thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-23 US disclosed
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090105253-A1 Triazole Derivative and Use Thereof F2R, HRH4, F2RL3 CCR1 184/4885ABCB1 1859/4885MLYCD 4763/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.