SCHEMBL5244366

SCHEMBL5244366

CCNC(=O)c1ccc(-n2nnc(C(=O)NCc3cccc(F)c3)c2CSC)cc1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.45
BRD4 O60885 1/20 0.44
LMNA P02545 2/20 0.43
MAPT P10636 2/20 0.42
ROCK2 O75116 2/20 0.42
TP53 P04637 1/20 0.42
NAMPT P43490 1/20 0.42
THRB P10828 1/20 0.42
GAA P10253 1/20 0.41
MMP13 P45452 1/20 0.41
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 1/20 0.40
RIPK1 Q13546 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5249308 0.92 RIPK1 (0.46) CCR1BRD4LMNAMAPTROCK2
SCHEMBL5248728 0.91 ABCB1 (0.47) BRD4LMNAMAPTTP53NAMPT
SCHEMBL3113720 0.91 CCR1 (0.43) CCR1BRD4LMNAMAPTROCK2
SCHEMBL5249263 0.91 LMNA (0.45) CCR1LMNAROCK2ALDH1A1
SCHEMBL3108441 0.90 CCR1 (0.47) CCR1BRD4LMNAMAPTROCK2
SCHEMBL5246361 0.89 CCR1 (0.49) CCR1LMNAMAPTROCK2THRB
SCHEMBL5246022 0.89 CCR1 (0.43) CCR1LMNAMAPTROCK2MEN1
SCHEMBL5248174 0.89 POLB (0.48) CCR1LMNAMAPTTP53THRB
SCHEMBL5244456 0.89 LMNA (0.57) LMNAMAPTALDH1A1
SCHEMBL5244694 0.89 HPGD (0.48) LMNAMAPTROCK2MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed