SCHEMBL3110491

SCHEMBL3110491

O=C(c1ccccc1)N1CC(O)C1

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.62
CHRNB4 P30926 2/20 0.62
CHRNA3 P32297 2/20 0.62
CHRNA7 P36544 2/20 0.62
CHRNA4 P43681 2/20 0.62
PLA2G1B P04054 1/20 0.57
ATG4B Q9Y4P1 1/20 0.57
HPGD P15428 2/20 0.57
ALDH1A1 P00352 2/20 0.56
ACHE P22303 1/20 0.55
SIGMAR1 Q99720 1/20 0.53
SLC18A3 Q16572 2/20 0.50
PIK3CD O00329 1/20 0.50
GRM5 P41594 1/20 0.50
EPHX1 P07099 1/20 0.50
USP2 O75604 1/20 0.50
L3MBTL3 Q96JM7 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
PDK2 Q15119 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8158994 0.89 HPGD (0.64) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL31360681 0.88 CHRNB2 (0.62) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL5871923 0.85 ACHE (0.62) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL2720515 0.85 ACHE (0.62) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL12442621 0.85 ACHE (0.62) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL3639020 0.84 GRM5 (0.73) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL11160146 0.84 CHRNB2 (0.59) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL28200535 0.82 HPGD (0.61) HPGDALDH1A1ACHESLC18A3USP2
SCHEMBL10274486 0.82 PLA2G1B (0.75) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL3650639 0.82 CHRNB2 (0.61) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025043225-A2 DEGRADERS OF CYCLIN-DEPENDENT KINASE 2 GENENTECH, INC. (US) 2025-02-27 WO disclosed
CN-117776997-A Preparation method of nitrogen-protected 3-hydroxy azetidine 风火轮(上海)生物科技有限公司 2024-03-29 CN disclosed
CN-111465602-B Synthesis of 4-aminopyrimidine compounds 帕劳制药有限公司 2023-05-23 CN disclosed
EP-3319955-B1 6-AMINO-QUINOLINE-3-CARBONITRILS AS COT MODULATORS GILEAD SCIENCES INC (US) 2020-11-25 EP disclosed
CN-111465602-A Synthesis of 4-aminopyrimidine compounds 森索睿翁公司 2020-07-28 CN disclosed
US-9920073-B2 Compositions useful for inhibiting HIV-1 infection and methods using same DREXEL UNIVERSITY (US) 2018-03-20 US disclosed
US-9920073-B2 Compositions useful for inhibiting HIV-1 infection and methods using same DREXEL UNIVERSITY (US) 2018-03-20 US disclosed
EP-2202223-B1 HETEROCYCLIC COMPOUND AS BLOOD RBP4 LOWERING AGENT TAKEDA PHARMACEUTICALS CO (JP) 2017-01-25 EP disclosed
EP-2202223-B1 HETEROCYCLIC COMPOUND AS BLOOD RBP4 LOWERING AGENT TAKEDA PHARMACEUTICALS CO (JP) 2017-01-25 EP disclosed
EP-2604597-B1 HETEROCYCLIC COMPOUND AND USE THEREOF INHIBITOR OF PHOSPHODIESTERASE 10A TAKEDA PHARMACEUTICALS CO (JP) 2017-01-04 EP disclosed
US-20140066420-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2014-03-06 US disclosed
US-8586571-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-11-19 US disclosed
US-8586571-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-11-19 US disclosed
EP-2604597-A1 HETEROCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2013-06-19 EP disclosed
US-20130137675-A1 HETEROCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-05-30 US disclosed
US-20100292206-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-11-18 US disclosed
US-20100292206-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-11-18 US disclosed
US-20100292206-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-11-18 US disclosed
EP-2202223-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2010-06-30 EP disclosed
US-4088644-A N-Acyl-3-azetidinone SCHERING-CORPORATION (US) 1978-05-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140066420-A1 HETEROCYCLIC COMPOUND RBP4, RBP1, RAVER1 CHRNB2 4113/4885CHRNB4 2264/4885CHRNA3 3404/4885
US-20130137675-A1 HETEROCYCLIC COMPOUND AND USE THEREOF PDE3A, PDE2A, PDE5A CHRNB2 553/4885CHRNB4 592/4885CHRNA3 357/4885
US-20100292206-A1 HETEROCYCLIC COMPOUND RBP4, RBP1, RAVER1 CHRNB2 4113/4885CHRNB4 2264/4885CHRNA3 3404/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.