SCHEMBL31107458

SCHEMBL31107458

C=C1C(=O)Nc2c(Br)cccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.42
CSNK1A1 P48729 1/20 0.42
CDK5 Q00535 1/20 0.42
ROCK1 Q13464 1/20 0.42
DYRK1A Q13627 1/20 0.42
LRRK2 Q5S007 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
DYRK1B Q9Y463 1/20 0.42
TGM2 P21980 1/20 0.42
PARP10 Q53GL7 1/20 0.40
PARP11 Q9NR21 1/20 0.40
PDE7A Q13946 5/20 0.39
DAO P14920 2/20 0.39
CES1 P23141 2/20 0.39
NSD2 O96028 1/20 0.39
BCHE P06276 1/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA7 P43166 2/20 0.39
CA9 Q16790 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29440762 0.80 CES1 (0.60) PIM1CSNK1A1CDK5ROCK1DYRK1A
SCHEMBL935810 0.80 CES1 (0.60) PIM1CSNK1A1CDK5ROCK1DYRK1A
SCHEMBL20535074 0.73 TGM2 (0.42) PIM1CSNK1A1CDK5ROCK1DYRK1A
SCHEMBL31107461 0.69 CES1 (0.43) PIM1CSNK1A1CDK5ROCK1DYRK1A
SCHEMBL15490689 0.69 GSK3B (0.71) LRRK2DYRK1BALDH1A1GSK3BPARP1
SCHEMBL13312397 0.68 GSK3B (0.41) PIM1CSNK1A1CDK5ROCK1DYRK1A
SCHEMBL22300869 0.67 MAOA (0.46) PIM1CSNK1A1CDK5ROCK1DYRK1A
SCHEMBL988494 0.67 LRRK2 (0.61) CDK5LRRK2DYRK1BTGM2ALDH1A1
SCHEMBL29479580 0.67 LRRK2 (0.61) CDK5LRRK2DYRK1BTGM2ALDH1A1
SCHEMBL7423435 0.67 CA1 (0.43) PIM1CSNK1A1CDK5ROCK1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118440081-A Four-ring condensed skeleton compound containing indoline unit and synthesis method thereof 西南交通大学 2024-08-06 CN claimed
CN-118440081-A Four-ring condensed skeleton compound containing indoline unit and synthesis method thereof 西南交通大学 2024-08-06 CN disclosed