SCHEMBL3120772

SCHEMBL3120772

CCCCOc1cc(N(Cc2cccnc2)c2cccc(C(=O)OC(=O)c3cccc(N(Cc4cncs4)c4ccc(OC(F)F)c(OCCCC)c4)c3)c2)ccc1OC(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 10/20 0.38
LMNA P02545 3/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
POLB P06746 2/20 0.34
MAPT P10636 2/20 0.34
PDE4B Q07343 2/20 0.34
KMT2A Q03164 1/20 0.34
NFKB1 P19838 2/20 0.34
NFKB2 Q00653 2/20 0.34
RELA Q04206 2/20 0.34
NPC1 O15118 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
JAK2 O60674 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3120759 0.94 GRM2 (0.40) GRM2PDE4BCYP3A4RXRA
SCHEMBL3129699 0.88 RXRA (0.42) LMNAPDE4BPDE4DRXRA
SCHEMBL3216620 0.87 HDAC6 (0.34) LMNAPDE4BPDE4APDE4CPDE4D
SCHEMBL3118000 0.87 GRM2 (0.44) GRM2LMNAPOLBMAPTPDE4B
SCHEMBL3201568 0.86 GRM2 (0.40) GRM2LMNAL3MBTL1CYP1A2CYP2C9
SCHEMBL3123568 0.84 ALDH1A1 (0.40) L3MBTL1CYP1A2TSHRCYP2C19POLB
SCHEMBL3132918 0.82 RXRA (0.45) GRM2TSHRPDE4BKMT2APDE4A
SCHEMBL3133648 0.82 RXRA (0.45) PDE4BPDE4DRXRA
SCHEMBL3133561 0.81 GRM2 (0.42) GRM2LMNAPOLBMAPTPDE4B
SCHEMBL3128993 0.80 HRH4 (0.39) LMNATSHRPOLBMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010003084-A2 PHOSPHODIESTERASE 4 INHIBITORS MEMORY PHARMACEUTICALS CORPORATION (US) 2010-01-07 WO disclosed