SCHEMBL312208

SCHEMBL312208

[O-][N+]1=Cc2ccccc2NC1

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11521800 0.61 GAA (0.32) GAAMAPT
SCHEMBL19679 0.61
SCHEMBL265188 0.60 MAOB (0.59)
SCHEMBL31337867 0.60 MAOB (0.59)
SCHEMBL8535074 0.58 GAA (0.37) GAAMAPT
SCHEMBL29415525 0.58 GAA (0.48) GAAMAPT
SCHEMBL34295 0.58 GAA (0.48) GAAMAPT
SCHEMBL160159 0.58 GAA (0.38) GAAMAPT
SCHEMBL2507520 0.57 GAA (0.36) GAAMAPT
Potassium SCHEMBL9683518 0.57 GAA (0.46) GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103524432-B One prepares the method for 2,3-dihydroquinazoline-4 (3H)-one analog derivative 贵州大学 2016-06-08 CN claimed
EP-2908817-A1 2,3-DIHYDROQUINAZOLIN-4(1 H)-ONE DERIVATIVES FOR USE IN THE TREATMENT OF VIRAL INFECTIONS Commissariat à l'Énergie Atomique et aux Énergies Alternatives (FR) 2015-08-26 EP claimed
WO-2014060588-A1 2,3-DIHYDROQUINAZOLIN-4(1 H)-ONE DERIVATIVES FOR USE IN THE TREATMENT OF VIRAL INFECTIONS COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2014-04-24 WO claimed
CN-103524432-A Method for preparing 2,3-dihydroquinazoline-4(3H)-ketone derivatives UNIV GUIZHOU 2014-01-22 CN claimed
EP-2350030-A1 ISOXAZOLE/ISOXAZOLINE/COMBRETASTATIN LINKED DIHYDROQUINAZOLINONE HYBRIDS AS POTENTIAL ANTICANCER AGENTS AND PROCESS FOR THE PREPARATION THEREOF Council Of Scientific & Industrial Research (IN) 2011-08-03 EP claimed
CN-101845021-A Quinazoline ketones alkaloid and preparation method and application thereof OCEAN UNIV CHINA 2010-09-29 CN claimed
WO-2010058417-A1 ISOXAZOLE/ISOXAZOLINE/COMBRETASTATIN LINKED DIHYDROQUINAZOLINONE HYBRIDS AS POTENTIAL ANTICANCER AGENTS AND PROCESS FOR THE PREPARATION THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2010-05-27 WO claimed
CN-104557737-B A kind of synthetic method of 2 aryl substituted quinazoline class medicine intermediates 王文明 2016-12-14 CN disclosed
CN-106083741-A 2 sulfur are for quinazolinedione derivatives 南京中医药大学 2016-11-09 CN disclosed
CN-103524432-B One prepares the method for 2,3-dihydroquinazoline-4 (3H)-one analog derivative 贵州大学 2016-06-08 CN disclosed
CN-104744380-A Method for preparing 2,3-dihydroquinazoline-4(1H)-one and derivative thereof UNIV ANHUI TECHNOLOGY 2015-07-01 CN disclosed
CN-104557737-A Method for synthesizing 2-aryl-substituted quinazoline medical intermediate MA LIANGJUN 2015-04-29 CN disclosed
CN-104356076-A Synthesis method for substituted 2, 3-dihydro-4(1H)-quinazolinone compound UNIV BOHAI 2015-02-18 CN disclosed
CN-1665804-A 4, 4-disubstituted piperidine derivatives having CCR3 antagonism TEIJIN LTD (JP) 2005-09-07 CN disclosed
EP-1507776-A1 2-OXO-1,3,4-TRIHYDROQUINAZOLINYL DERIVATIVES FOR THE TREATMENT OF CELL PROLIFERATION-RELATED DISORDERS Amgen Inc. (US) 2005-02-23 EP disclosed
CN-1578768-A Anthranilamides and pharmaceutical use thereof NOVARTIS AG (CH) 2005-02-09 CN disclosed
US-20030232846-A1 Caspase inhibitors and uses thereof VERTEX PHARMACEUTICALS INCORPORATED 2003-12-18 US disclosed
WO-2003101985-A1 2-OXO-1,3,4-TRIHYDROQUINAZOLINYL DERIVATIVES FOR THE TREATMENT OF CELL PROLIFERATION-RELATED DISORDERS AMGEN INC. (US) 2003-12-11 WO disclosed
EP-1244626-A2 CASPASE INHIBITORS AND USES THEREOF Vertex Pharmaceuticals Incorporated (US) 2002-10-02 EP disclosed
WO-2001042216-A2 CASPASE INHIBITORS AND USES THEREOF VERTEX PHARMACEUTICALS INCORPORATED (US) 2001-06-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030232846-A1 Caspase inhibitors and uses thereof CASP1, CASP3, CASP2 GAA 2029/4885MAPT 3562/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.