SCHEMBL31228005

SCHEMBL31228005

Cc1cnc2[nH]cc(I)c2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.54
CYP2C9 P11712 6/20 0.43
CYP2C19 P33261 4/20 0.43
CYP3A4 P08684 7/20 0.41
MAPK1 P28482 1/20 0.41
AXL P30530 1/20 0.38
CDK8 P49336 1/20 0.38
TNIK Q9UKE5 1/20 0.38
KIT P10721 1/20 0.38
DYRK1A Q13627 2/20 0.36
PLK4 O00444 1/20 0.36
AURKA O14965 1/20 0.36
JAK2 O60674 1/20 0.36
ROCK2 O75116 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
PRKCG P05129 1/20 0.36
INSR P06213 1/20 0.36
CDK1 P06493 1/20 0.36
FES P07332 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1045946 1.00 BRD4 (0.54) BRD4CYP2C9CYP2C19CYP3A4MAPK1
SCHEMBL15241762 0.80 BRD4 (0.49) BRD4MAPK1AXLCDK8TNIK
SCHEMBL7921128 0.80 MET (0.46) CYP2C9CYP2C19CYP3A4AXLITK
SCHEMBL25971496 0.77 BRD4 (0.47) BRD4MAPK1AXLCDK8TNIK
SCHEMBL1053943 0.77 JAK2 (0.58) BRD4CYP2C9CYP2C19CYP3A4MAPK1
SCHEMBL7912970 0.77 BRD4 (0.47) BRD4MAPK1AXLCDK8TNIK
SCHEMBL1880862 0.77 BRD4 (0.47) BRD4MAPK1AXLCDK8TNIK
SCHEMBL68662 0.77 DYRK1A (0.58) BRD4MAPK1AXLCDK8TNIK
SCHEMBL11968454 0.77 BRD4 (0.47) BRD4MAPK1AXLCDK8TNIK
SCHEMBL13199598 0.77 CYP3A4 (0.44) CYP2C9CYP2C19CYP3A4KITKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119431362-A Substituted heteroaryl carboxylic acid compound, preparation method and pharmaceutical application thereof 中国医学科学院药物研究所 2025-02-14 CN disclosed
CN-118772152-A Azacyclic compounds as AAK1 inhibitors 艾立康药业股份有限公司 2024-10-15 CN disclosed