SCHEMBL3122986

SCHEMBL3122986

N#Cc1ccc(-c2cnn(C3CC[N]CC3)c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 4/20 0.47
MAP3K7 O43318 1/20 0.41
TAB1 Q15750 1/20 0.41
CCNA2 P20248 2/20 0.40
CDK2 P24941 2/20 0.40
CCNK O75909 2/20 0.40
CDK12 Q9NYV4 2/20 0.40
EP300 Q09472 2/20 0.40
PIK3CD O00329 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
PI4KA P42356 1/20 0.40
PIK3CG P48736 1/20 0.40
PI4KB Q9UBF8 1/20 0.40
KDM1A O60341 1/20 0.39
PAK1 Q13153 2/20 0.39
MAP4K3 Q8IVH8 1/20 0.38
IRAK4 Q9NWZ3 2/20 0.37
IRAK1 P51617 1/20 0.37
CREBBP Q92793 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3246673 0.81 RIPK1 (0.46) ALKPIK3CDPIK3CAPIK3CBPI4KA
SCHEMBL3124619 0.81 MAP4K3 (0.46) PIK3CDPIK3CAPIK3CBPI4KAPIK3CG
SCHEMBL2299419 0.80 CHRNB2 (0.47) ALKMAP3K7TAB1PIK3CDPIK3CA
SCHEMBL3118153 0.77 MAP4K3 (0.48) PIK3CDPIK3CAPIK3CBPI4KAPIK3CG
SCHEMBL3118417 0.77 ALK (0.49) ALKCDK2PIK3CDPIK3CAPIK3CB
SCHEMBL30440960 0.76 ALK (0.46) ALKMAP3K7TAB1CCNA2CDK2
SCHEMBL27030554 0.76 ALK (0.45) ALKMAP3K7TAB1EP300PIK3CD
SCHEMBL25424497 0.75 KDR (0.47) ALKMAP3K7TAB1KDM1AIRAK4
SCHEMBL3247635 0.72 PIK3CD (0.40) MAP3K7TAB1PIK3CDPIK3CAPIK3CB
SCHEMBL27030656 0.72 ALK (0.48) ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010022055-A2 INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS AMGEN INC. (US) 2010-02-25 WO disclosed