SCHEMBL3126331

SCHEMBL3126331

N#Cc1ccccc1-c1ccc(Br)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.66
PTGES O14684 2/20 0.59
PTPN5 P54829 1/20 0.50
LMNA P02545 1/20 0.46
TRPA1 O75762 1/20 0.45
ALDH1A1 P00352 4/20 0.44
MAPK1 P28482 2/20 0.44
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA5 P31644 1/20 0.44
GABRA3 P34903 1/20 0.44
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
HSD17B10 Q99714 2/20 0.43
CLK4 Q9HAZ1 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
ALOX5AP P20292 1/20 0.42
FEN1 P39748 1/20 0.42
AGTR1 P30556 1/20 0.41
ADORA2A P29274 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31410710 0.87 ESR2 (0.76) ESR2PTGESPTPN5TRPA1ALDH1A1
SCHEMBL2016996 0.83 ESR2 (0.70) ESR2PTGESPTPN5TRPA1ALDH1A1
SCHEMBL3947197 0.83 ALDH1A1 (0.48) ESR2PTGESPTPN5LMNAALDH1A1
Water SCHEMBL3178714 0.82 ESR2 (0.69) ESR2PTPN5TRPA1ALDH1A1GABRG2
SCHEMBL27895577 0.82 ESR2 (0.69) ESR2PTGESPTPN5TRPA1ALDH1A1
SCHEMBL29662886 0.82 ESR2 (0.69) ESR2PTPN5TRPA1ALDH1A1GABRG2
SCHEMBL223 0.82 ESR2 (0.69) ESR2PTPN5TRPA1ALDH1A1GABRG2
SCHEMBL18411231 0.82 ESR2 (0.53) ESR2PTGESPTPN5LMNATRPA1
SCHEMBL28571074 0.81 ESR2 (0.68) ESR2PTGESPTPN5TRPA1ALDH1A1
SCHEMBL151224 0.80 ESR2 (0.67) ESR2PTPN5LMNATRPA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112745318-B Compound and application thereof 北京鼎材科技有限公司 2024-03-19 CN disclosed
CN-112778300-B Organic compound and organic electroluminescent device containing the same 北京鼎材科技有限公司 2024-02-02 CN disclosed
CN-115894472-A Preparation method of high-purity azilsartan medoxomil potassium salt 仁合益康集团有限公司 2023-04-04 CN disclosed
US-20180212158-A1 ORGANIC LIGHT-EMITTING DIODE MATERIALS PRESIDENT AND FELLOWS OF HARVARD COLLEGE 2018-07-26 US disclosed
US-20180212158-A1 ORGANIC LIGHT-EMITTING DIODE MATERIALS PRESIDENT AND FELLOWS OF HARVARD COLLEGE 2018-07-26 US disclosed
WO-2017011531-A2 ORGANIC LIGHT-EMITTING DIODE MATERIALS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2017-01-19 WO disclosed
US-7642361-B2 Thiophene and furan compounds ELI LILLY AND COMPANY (US) 2010-01-05 US disclosed
US-7642361-B2 Thiophene and furan compounds ELI LILLY AND COMPANY (US) 2010-01-05 US disclosed
US-7642361-B2 Thiophene and furan compounds ELI LILLY AND COMPANY (US) 2010-01-05 US disclosed
US-7625932-B2 Pyrrole and pyrazole derivatives as potentiators of glutamate receptors ELI LILLY AND COMPANY (US) 2009-12-01 US disclosed
US-20070105852-A1 Thiophene and furan compounds ELI LILLY AND COMPANY 2007-05-10 US disclosed
US-20070066573-A1 Pyrrole and pyrazole derivatives as potentiators of glutamate receptors ELI LILLY AND COMPANY 2007-03-22 US disclosed
US-20070066573-A1 Pyrrole and pyrazole derivatives as potentiators of glutamate receptors ELI LILLY AND COMPANY 2007-03-22 US disclosed
US-20070066573-A1 Pyrrole and pyrazole derivatives as potentiators of glutamate receptors ELI LILLY AND COMPANY 2007-03-22 US disclosed
EP-1706395-A1 THIOPHENE AND FURAN COMPOUNDS ELI LILLY AND COMPANY (US) 2006-10-04 EP disclosed
EP-1670757-A1 PYRROLE AND PYRAZOLE DERIVATIVES AS POTENTIATORS OF GLUTAMATE RECEPTORS ELI LILLY AND COMPANY (US) 2006-06-21 EP disclosed
WO-2005070916-A1 THIOPHENE AND FURAN COMPOUNDS ELI LILLY AND COMPANY (US) 2005-08-04 WO disclosed
WO-2005070916-A1 THIOPHENE AND FURAN COMPOUNDS ELI LILLY AND COMPANY (US) 2005-08-04 WO disclosed
WO-2005040110-A1 PYRROLE AND PYRAZOLE DERIVATIVES AS POTENTIATORS OF GLUTAMATE RECEPTORS ELI LILLY AND COMPANY (US) 2005-05-06 WO disclosed
WO-2005040110-A1 PYRROLE AND PYRAZOLE DERIVATIVES AS POTENTIATORS OF GLUTAMATE RECEPTORS ELI LILLY AND COMPANY (US) 2005-05-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180212158-A1 ORGANIC LIGHT-EMITTING DIODE MATERIALS MSN, DDT, NECTIN4 ESR2 382/4885PTGES 2447/4885PTPN5 4155/4885
US-20070105852-A1 Thiophene and furan compounds PSEN2, PSEN1, TPMT ESR2 1593/4885PTGES 625/4885PTPN5 805/4885
US-20070066573-A1 Pyrrole and pyrazole derivatives as potentiators of glutamate receptors GRIN1, GRIN3A, GRIK5 ESR2 706/4885PTGES 1479/4885PTPN5 2380/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.