SCHEMBL3396593

SCHEMBL3396593

COc1ccc(-c2cnnc(N)n2)c(C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.45
HSP90AA1 P07900 2/20 0.42
HSP90AB1 P08238 2/20 0.42
CRHR1 P34998 2/20 0.40
NPC1 O15118 1/20 0.40
ACHE P22303 1/20 0.39
MAPT P10636 3/20 0.38
ALDH1A1 P00352 2/20 0.38
HTT P42858 2/20 0.38
LIMK1 P53667 2/20 0.38
DYRK1A Q13627 1/20 0.38
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
KPNA2 P52292 1/20 0.37
EIF4E P06730 1/20 0.37
SCN9A Q15858 1/20 0.37
TP53 P04637 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13425829 0.83 ADORA2A (0.39) KDM4EGLAGAASCN9ATSHR
SCHEMBL3395686 0.80 HSD17B1 (0.40) KDM4ENPC1MAPTALDH1A1GLA
SCHEMBL3395005 0.78 DHFR (0.47) KDM4EHSP90AA1HSP90AB1NPC1MAPT
SCHEMBL3394338 0.76 AR (0.41) GLAGAASCN9ATSHRADORA2A
SCHEMBL3128136 0.76 ATR (0.48) ADORA2AADORA1
SCHEMBL3399081 0.73 ADORA2A (0.51) KDM4ENPC1DYRK1AADORA2AADORA1
SCHEMBL19436331 0.73 ADORA2A (0.60) KDM4EACHEADORA2AADORA1
SCHEMBL4049824 0.72 CRHR1 (0.40) CRHR1NPC1MAPTLIMK1EIF4E
SCHEMBL2324238 0.72 ADORA2A (0.62) KDM4ENPC1MAPTALDH1A1HTT
SCHEMBL2322961 0.71 ADORA2A (0.50) KDM4ENPC1MAPTALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed