SCHEMBL312905

SCHEMBL312905

C[C](C)c1ccc(CNC(=O)c2cc(-c3ccccc3)oc2C)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.52
MEN1 O00255 6/20 0.52
KMT2A Q03164 6/20 0.52
HPGD P15428 4/20 0.52
LMNA P02545 2/20 0.52
L3MBTL1 Q9Y468 2/20 0.52
KDM4E B2RXH2 1/20 0.52
MAPT P10636 3/20 0.50
CYP1A2 P05177 2/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
CYP2D6 P10635 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
ALOX12 P18054 1/20 0.50
PKM P14618 1/20 0.49
HTT P42858 1/20 0.49
HSD17B10 Q99714 1/20 0.49
NPSR1 Q6W5P4 1/20 0.47
ALPL P05186 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25910313 0.91 ALDH1A1 (0.53) ALDH1A1MEN1KMT2AHPGDLMNA
SCHEMBL8230805 0.87 KLKB1 (0.57) ALDH1A1MEN1KMT2AHPGDLMNA
SCHEMBL313244 0.81 ALDH1A1 (0.73) ALDH1A1MEN1KMT2AHPGDLMNA
SCHEMBL13753348 0.79 ALDH1A1 (0.59) ALDH1A1MEN1KMT2AHPGDLMNA
SCHEMBL8507040 0.78 ALDH1A1 (0.63) ALDH1A1MEN1KMT2AHPGDLMNA
SCHEMBL2695793 0.76 CCR2 (0.56) ALDH1A1HPGDLMNAL3MBTL1KDM4E
Hydrochloric Acid SCHEMBL2907820 0.76 CCR2 (0.55) ALDH1A1HPGDLMNAL3MBTL1KDM4E
Iodide SCHEMBL17555122 0.76 CCR2 (0.55) ALDH1A1HPGDLMNAL3MBTL1KDM4E
SCHEMBL14434229 0.73 KDM4E (0.57) ALDH1A1MEN1KMT2AHPGDLMNA
SCHEMBL9834670 0.73 ALDH1A1 (0.59) ALDH1A1MEN1KMT2AHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093428-B2 Synthesis of quaternary salt compounds JANSSEN PHARMACEUTICA N.V. (BE) 2012-01-10 US disclosed