SCHEMBL3129372

SCHEMBL3129372

COc1cccc(CNC(=O)Nc2ccc(-c3ccnc4[nH]cnc34)cc2OCCCO)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 9/20 0.47
F3 P13726 1/20 0.44
ROCK1 Q13464 4/20 0.43
ALDH1A1 P00352 2/20 0.42
CIT O14578 1/20 0.42
TNIK Q9UKE5 1/20 0.42
DGAT2 Q96PD7 2/20 0.41
KMT2A Q03164 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP3A5 P20815 1/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41
GFER P55789 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
PRKACA P17612 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3244785 0.88 CIT (0.57) ROCK2F3ROCK1CITTNIK
SCHEMBL3244355 0.85 ROCK2 (0.53) ROCK2F3ROCK1ALDH1A1CIT
SCHEMBL3240812 0.82 ROCK2 (0.51) ROCK2F3ROCK1ALDH1A1KMT2A
SCHEMBL13391340 0.80 ROCK2 (0.67) ROCK2ROCK1PRKACA
SCHEMBL3130579 0.78 JAK3 (0.47) ROCK2ROCK1ALDH1A1CITTNIK
SCHEMBL3245171 0.77 ROCK2 (0.69) ROCK2ROCK1PRKACA
SCHEMBL3239562 0.73 ROCK2 (0.59) ROCK2ROCK1
SCHEMBL3245457 0.73 ROCK2 (0.68) ROCK2ROCK1PRKACA
SCHEMBL3243730 0.73 ROCK2 (0.58) ROCK2ROCK1CITTNIKCYP3A4
SCHEMBL3242171 0.72 ROCK2 (0.67) ROCK2ROCK1PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO claimed
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO disclosed