SCHEMBL3244785

SCHEMBL3244785

COc1cccc(CNC(=O)Nc2ccc(-c3ccnc4[nH]ccc34)cc2OCCCO)c1

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CIT O14578 4/20 0.57
TNIK Q9UKE5 2/20 0.49
ROCK2 O75116 8/20 0.48
ROCK1 Q13464 3/20 0.48
BRAF P15056 2/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
F3 P13726 1/20 0.44
DGAT2 Q96PD7 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3244355 0.88 ROCK2 (0.53) CITROCK2ROCK1F3DGAT2
SCHEMBL3129372 0.88 ROCK2 (0.47) CITTNIKROCK2ROCK1CYP2D6
SCHEMBL3130579 0.88 JAK3 (0.47) CITTNIKROCK2ROCK1
SCHEMBL3243730 0.85 ROCK2 (0.58) CITTNIKROCK2ROCK1BRAF
SCHEMBL3248895 0.83 ROCK2 (0.55) CITTNIKROCK2ROCK1BRAF
SCHEMBL3240812 0.82 ROCK2 (0.51) ROCK2ROCK1F3
SCHEMBL13391340 0.80 ROCK2 (0.67) ROCK2ROCK1
SCHEMBL3245171 0.77 ROCK2 (0.69) ROCK2ROCK1
SCHEMBL1647246 0.74 PRKACA (0.65) CITTNIKROCK2ROCK1CYP2D6
SCHEMBL12779735 0.74 ROCK2 (0.70) CITTNIKROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO claimed
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO disclosed