SCHEMBL3130169

SCHEMBL3130169

CCCc1ccnc2[nH]cc(-c3ccnc(Nc4cccc(S(N)(=O)=O)c4)n3)c12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 16/20 0.59
MTOR P42345 8/20 0.59
SMG1 Q96Q15 7/20 0.59
SLC2A1 P11166 1/20 0.52
CDK2 P24941 11/20 0.52
CDK9 P50750 9/20 0.52
CCNB1 P14635 9/20 0.52
CCNT1 O60563 8/20 0.52
CCNA2 P20248 5/20 0.51
CDK7 P50613 5/20 0.51
CCNH P51946 5/20 0.51
CCNA1 P78396 5/20 0.51
PIK3CA P42336 1/20 0.51
PIK3CG P48736 1/20 0.51
IKBKB O14920 1/20 0.49
AURKA O14965 1/20 0.46
MAP4K4 O95819 1/20 0.46
ABL1 P00519 1/20 0.46
LCK P06239 1/20 0.46
MET P08581 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3623836 0.77 CDK1 (0.55) CDK1MTORSMG1SLC2A1CDK2
SCHEMBL3132734 0.74 IKBKB (0.49) CDK1CDK2CDK9CCNB1CCNT1
SCHEMBL6752979 0.74 CAMK2D (0.67) CDK1MTORSMG1SLC2A1CDK2
SCHEMBL7524252 0.74 CDK1 (0.69) CDK1MTORSMG1SLC2A1CDK2
SCHEMBL2988085 0.73 CDK5 (0.67) CDK1CDK2CDK9CCNB1CCNT1
SCHEMBL3518683 0.73 IKBKB (0.66) CDK1MTORSMG1SLC2A1CDK2
SCHEMBL7471938 0.73 ABL1 (0.70) CDK1MTORSMG1SLC2A1CDK2
SCHEMBL3607096 0.72 CDK9 (0.62) CDK1MTORSMG1SLC2A1CDK2
SCHEMBL3520990 0.72 CDK1 (0.66) CDK1MTORSMG1SLC2A1CDK2
SCHEMBL3623043 0.72 KDR (0.63) CDK1MTORSMG1SLC2A1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010051781-A1 KINASE INHIBITORS AND THEIR USE AS PHARMACEUTICAL AGENTS SHANGHAI GENOMICS, INC. (CN) 2010-05-14 WO disclosed