SCHEMBL3130951

SCHEMBL3130951

O=C(CN1C(=O)CCc2cc(-c3cc(Cl)cc(Cl)c3)cnc21)N1CCc2ccc(O)cc2C1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.43
ESR2 Q92731 4/20 0.43
MAPK1 P28482 10/20 0.39
ALDH1A1 P00352 1/20 0.36
ERCC1 P07992 1/20 0.36
ERCC4 Q92889 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GAA P10253 1/20 0.36
TSHR P16473 1/20 0.36
CYP11B2 P19099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3267887 0.92 MAPK1 (0.45) MAPK1ALDH1A1KDM4ELMNAHTT
SCHEMBL3127545 0.90 MAPK1 (0.41) ESR1ESR2MAPK1ALDH1A1KDM4E
SCHEMBL3118590 0.86 ESR2 (0.45) ESR1ESR2MAPK1ALDH1A1KDM4E
SCHEMBL3246493 0.85 FNTA (0.39) MAPK1ALDH1A1KDM4ELMNAHTT
SCHEMBL3264528 0.83 MAPK1 (0.44) ESR1ESR2MAPK1ALDH1A1KDM4E
SCHEMBL13521598 0.82 HSD17B3 (0.43) ESR1ESR2MAPK1ALDH1A1KDM4E
SCHEMBL3251252 0.82 GAA (0.47) ESR1ESR2MAPK1ALDH1A1KDM4E
SCHEMBL3124617 0.79 GRIN2B (0.42) ESR1ESR2MAPK1
SCHEMBL3241068 0.79 CYP11B2 (0.41) CYP11B2
SCHEMBL3119024 0.79 TAAR1 (0.46) ESR1ESR2MAPK1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO claimed