SCHEMBL31335544

SCHEMBL31335544

C=CC(=O)N(C)c1ccc2c(n1)CN(C(=O)c1c(O)cc(OC)c(Cl)c1C)CC2

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 5/20 0.38
FGFR4 P22455 5/20 0.38
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
FGFR2 P21802 1/20 0.34
FGFR3 P22607 1/20 0.34
SPR P35270 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
KRAS P01116 4/20 0.34
MAPK1 P28482 1/20 0.33
ABCB1 P08183 1/20 0.32
LMNA P02545 1/20 0.32
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31335683 0.91 KMT2A (0.34) KMT2AMEN1SPRCA1CA2
SCHEMBL31335613 0.87 FGFR1 (0.38) FGFR1FGFR4KMT2AMEN1SPR
SCHEMBL31335590 0.84 FGFR1 (0.41) FGFR1FGFR4KMT2AMEN1FGFR2
SCHEMBL31335742 0.84 SPR (0.39) FGFR1FGFR4KMT2AMEN1SPR
SCHEMBL31335773 0.84 FGFR4 (0.39) FGFR1FGFR4KMT2AMEN1SPR
SCHEMBL31335782 0.77 FGFR1 (0.37) FGFR1FGFR4KMT2AMEN1FGFR2
SCHEMBL31335632 0.76 MAPT (0.39) KMT2AMEN1CA1CA2CA7
SCHEMBL31335690 0.75 SPR (0.39) KMT2AMEN1SPRCA1CA2
SCHEMBL31335751 0.75 TRAP1 (0.40) FGFR1FGFR4SPRKRAS
SCHEMBL31335490 0.74 SPR (0.42) KMT2AMEN1SPRCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4720038-A1 (HETERO)ARYL-CARBONYL-HETEROBICYCLIC COMPOUNDS AS INHIBITORS OF PMS2 FOR CANCER AND DEGENERATIVE ILLNESSES Neophore Limited (GB) 2026-04-08 EP claimed
WO-2024246496-A1 (HETERO)ARYL-CARBONYL-HETEROBICYCLIC COMPOUNDS AS INHIBITORS OF PMS2 FOR CANCER AND DEGENERATIVE ILLNESSES Neophore Limited (GB) 2024-12-05 WO claimed
EP-4720038-A1 (HETERO)ARYL-CARBONYL-HETEROBICYCLIC COMPOUNDS AS INHIBITORS OF PMS2 FOR CANCER AND DEGENERATIVE ILLNESSES Neophore Limited (GB) 2026-04-08 EP disclosed
WO-2024246496-A1 (HETERO)ARYL-CARBONYL-HETEROBICYCLIC COMPOUNDS AS INHIBITORS OF PMS2 FOR CANCER AND DEGENERATIVE ILLNESSES Neophore Limited (GB) 2024-12-05 WO disclosed