SCHEMBL31455019

SCHEMBL31455019

COC(=O)C1CC2(CC(C(=O)Nc3ccc(Nc4nc(-c5ccccc5)ccc4[N+](=O)[O-])c(C)n3)C2)C1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
ADORA1 P30542 8/20 0.33
ADORA2A P29274 6/20 0.33
ADORA3 P0DMS8 5/20 0.33
ABCB1 P08183 6/20 0.33
ABCC1 P33527 3/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31455406 0.94 CYP3A4 (0.34) GSK3AGSK3BADORA1ADORA2AADORA3
SCHEMBL31455204 0.89 GSK3B (0.38) GSK3AGSK3BADORA1ADORA2AADORA3
SCHEMBL31455141 0.87 POLB (0.36) ABCB1ABCC1NPC1
SCHEMBL31455145 0.87 CYP3A4 (0.33) GSK3AGSK3BADORA1ADORA2AADORA3
SCHEMBL31455274 0.87 HDAC1 (0.38) GSK3AGSK3BADORA1ADORA2AADORA3
SCHEMBL31455069 0.85 GSK3A (0.35) GSK3AGSK3BADORA1ADORA2AADORA3
SCHEMBL31455487 0.82 HDAC1 (0.36) GSK3AGSK3BADORA1ADORA2AADORA3
SCHEMBL31455449 0.79 GSK3B (0.39) GSK3AGSK3BADORA1ADORA2AADORA3
SCHEMBL31455361 0.79 ADORA1 (0.40) GSK3AGSK3BADORA1ADORA2AADORA3
SCHEMBL31455065 0.78 ABCB1 (0.44) GSK3BADORA1ADORA2AADORA3ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025059577-A1 SUBSTITUTED AMINOPYRIDINE COMPOUNDS FOR USE AS AKT1 INHIBITORS ATAVISTIK BIO, INC. (US) 2025-03-20 WO disclosed