SCHEMBL3145780

SCHEMBL3145780

CN(C(=O)O)C1(CNc2cnc(Cl)c(-c3ccc(N)cc3)c2)CC1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 4/20 0.34
FFAR4 Q5NUL3 5/20 0.33
CCNT1 O60563 3/20 0.33
CDK9 P50750 3/20 0.33
CDK2 P24941 1/20 0.33
USP28 Q96RU2 1/20 0.32
CLK1 P49759 1/20 0.31
DYRK1A Q13627 1/20 0.31
FNTA P49354 2/20 0.31
FNTB P49356 2/20 0.31
PGGT1B P53609 1/20 0.31
ATM Q13315 1/20 0.31
CYP1A2 P05177 1/20 0.30
GSK3B P49841 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3146191 0.92 MAP4K4 (0.37) MAP4K4FFAR4CCNT1CDK9CDK2
SCHEMBL3143345 0.89 CYP46A1 (0.35) CCNT1CDK9CDK2FNTAFNTB
SCHEMBL3147370 0.89 ABL1 (0.36) CLK1DYRK1AATM
SCHEMBL3152381 0.87 AR (0.38) MAP4K4
SCHEMBL3770604 0.81 FFAR4 (0.33) MAP4K4FFAR4CCNT1CDK9CDK2
SCHEMBL3257000 0.80 FFAR4 (0.42) MAP4K4FFAR4
SCHEMBL3156239 0.79 ALDH1A1 (0.33)
SCHEMBL3141366 0.77 SYK (0.37) CCNT1CDK9CDK2CLK1DYRK1A
SCHEMBL3151064 0.77 RAF1 (0.38)
Hydrochloric Acid SCHEMBL3778971 0.76 SYK (0.36) MAP4K4CCNT1CDK9CDK2CLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed