SCHEMBL3146191

SCHEMBL3146191

CN(C(=O)O)C1(CNc2cnc(Cl)c(-c3ccc(Cl)cc3)c2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 4/20 0.37
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA7 P36544 1/20 0.36
MALT1 Q9UDY8 2/20 0.34
EGLN1 Q9GZT9 2/20 0.33
CCNT1 O60563 1/20 0.33
CDK2 P24941 1/20 0.33
CDK9 P50750 1/20 0.33
GPR119 Q8TDV5 2/20 0.33
DGAT1 O75907 1/20 0.33
KCNH2 Q12809 1/20 0.33
RAB9A P51151 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
KDM4E B2RXH2 2/20 0.33
NPC1 O15118 2/20 0.33
MAPT P10636 2/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3145780 0.92 MAP4K4 (0.34) MAP4K4CCNT1CDK2CDK9FFAR4
SCHEMBL3143345 0.91 CYP46A1 (0.35) CCNT1CDK2CDK9
SCHEMBL3152381 0.89 AR (0.38) MAP4K4EGLN1GPR119EGLN3CNR1
SCHEMBL3156239 0.81 ALDH1A1 (0.33) KCNH2MAPTLMNAALDH1A1
SCHEMBL3147370 0.80 ABL1 (0.36) KCNH2
SCHEMBL3771958 0.80 MAP4K4 (0.35) MAP4K4CHRNB4CHRNA3CHRNA7MALT1
SCHEMBL3146681 0.80 CHRNB4 (0.45) MAP4K4CHRNB4CHRNA3CHRNA7KCNH2
SCHEMBL3151064 0.79 RAF1 (0.38)
SCHEMBL3146187 0.78 MAP4K4 (0.38) MAP4K4CHRNB4CHRNA3CHRNA7MALT1
SCHEMBL4818195 0.77 KCNQ3 (0.41) RAB9ASMN1; SMN2MAPTLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed