SCHEMBL3145987

SCHEMBL3145987

CCc1ccc(-c2cncc(OCC3(CN)CC3)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 2/20 0.40
BACE1 P56817 1/20 0.37
KCNH2 Q12809 1/20 0.37
PRMT5 O14744 1/20 0.37
WDR77 Q9BQA1 1/20 0.37
CHRNB2 P17787 7/20 0.37
CHRNB1 P11230 6/20 0.37
CHRNB4 P30926 6/20 0.37
CHRNA3 P32297 6/20 0.37
CHRNB3 Q05901 6/20 0.37
AKT1 P31749 2/20 0.37
CDC7 O00311 1/20 0.37
DAPK3 O43293 1/20 0.37
DYRK3 O43781 1/20 0.37
ROCK2 O75116 1/20 0.37
RPS6KA5 O75582 1/20 0.37
PRKD3 O94806 1/20 0.37
MAP4K4 O95819 1/20 0.37
PRKCG P05129 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3785911 0.99 CYP11B1 (0.39) CYP11B1CYP11B2BACE1KCNH2PRMT5
SCHEMBL3137051 0.86 CHRNB1 (0.49) CYP11B1CYP11B2BACE1KCNH2PRMT5
Hydrochloric Acid SCHEMBL3145821 0.85 CHRNB1 (0.48) CYP11B1CYP11B2BACE1KCNH2PRMT5
SCHEMBL3137136 0.85 CHRNB2 (0.47) CYP11B1CYP11B2PRMT5WDR77CHRNB2
SCHEMBL3145265 0.85 CHRNB2 (0.47) CYP11B1CYP11B2BACE1KCNH2PRMT5
Hydrochloric Acid SCHEMBL3146592 0.84 CHRNB2 (0.46) CYP11B1CYP11B2BACE1KCNH2PRMT5
Hydrochloric Acid SCHEMBL3773007 0.84 CHRNB2 (0.46) CYP11B1CYP11B2BACE1KCNH2PRMT5
Hydrochloric Acid SCHEMBL3780020 0.84 CHRNB2 (0.46) CYP11B1CYP11B2PRMT5WDR77CHRNB2
SCHEMBL3150643 0.81 MKNK1 (0.41) CYP11B1CYP11B2CHRNB2CHRNB1CHRNB4
SCHEMBL3145991 0.80 CYP11B1 (0.40) CYP11B1CYP11B2BACE1KCNH2CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed