SCHEMBL3146709

SCHEMBL3146709

NCC1(COc2cnc(F)c(-c3cccc(Cl)c3)c2)CC1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
DHFR P00374 1/20 0.37
HRH1 P35367 1/20 0.36
TDO2 P48775 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
BACE1 P56817 1/20 0.34
KCNH2 Q12809 1/20 0.34
KDM1A O60341 1/20 0.34
MAOB P27338 1/20 0.34
DPP4 P27487 1/20 0.33
PTPN11 Q06124 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3774047 0.99 CHRNB2 (0.41) CHRNB2CHRNA4DHFRHRH1TDO2
Hydrochloric Acid SCHEMBL3770716 0.99 CHRNB2 (0.41) CHRNB2CHRNA4DHFRHRH1TDO2
SCHEMBL3145347 0.89 DHFR (0.37) DHFRHRH1TDO2ADORA2AADORA1
SCHEMBL3155932 0.88 DHFR (0.39) DHFRHRH1TDO2ADORA2AADORA1
Hydrochloric Acid SCHEMBL3773421 0.88 DHFR (0.36) DHFRHRH1TDO2ADORA2AADORA1
SCHEMBL3155137 0.87 MAP4K4 (0.35) CHRNB2
Hydrochloric Acid SCHEMBL3767963 0.87 DHFR (0.38) DHFRHRH1TDO2ADORA2AADORA1
SCHEMBL3143008 0.87 CHRNB4 (0.39) BACE1KCNH2KDM1A
Hydrochloric Acid SCHEMBL3770439 0.86 MAP4K4 (0.35) CHRNB2
Hydrochloric Acid SCHEMBL3773488 0.86 CHRNB4 (0.39) BACE1KCNH2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed