SCHEMBL3155137

SCHEMBL3155137

NCC1(COc2cnc(F)c(-c3cccc(N)c3)c2)CC1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 3/20 0.35
FYN P06241 1/20 0.35
CHRNB1 P11230 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNB3 Q05901 1/20 0.35
KIT P10721 3/20 0.33
CLK1 P49759 1/20 0.33
DYRK1A Q13627 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3770439 0.99 MAP4K4 (0.35) MAP4K4FYNCHRNB1CHRNB2CHRNB4
SCHEMBL3144019 0.88 FYN (0.37) MAP4K4FYNCHRNB1CHRNB2CHRNB4
Hydrochloric Acid SCHEMBL3768581 0.87 FYN (0.37) MAP4K4FYNCHRNB1CHRNB2CHRNB4
SCHEMBL3146709 0.87 CHRNB2 (0.41) CHRNB2
SCHEMBL3150790 0.87 PRKCZ (0.32)
Hydrochloric Acid SCHEMBL3774047 0.86 CHRNB2 (0.41) CHRNB2
Hydrochloric Acid SCHEMBL3770716 0.86 CHRNB2 (0.41) CHRNB2
SCHEMBL3154920 0.86 MAP4K4 (0.35) MAP4K4FYNCHRNB4CHRNA3
Hydrochloric Acid SCHEMBL3774548 0.86 PRKCZ (0.32)
Hydrochloric Acid SCHEMBL3776437 0.85 MAP4K4 (0.35) MAP4K4FYNCHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed