SCHEMBL3147201

SCHEMBL3147201

CNC1(COc2cncc(-c3ccc(SC)cc3)c2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
INPPL1 O15357 1/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
CHRNB2 P17787 5/20 0.36
CHRNB1 P11230 4/20 0.36
CHRNB4 P30926 4/20 0.36
CHRNA3 P32297 4/20 0.36
CHRNB3 Q05901 4/20 0.36
CHRNA4 P43681 1/20 0.35
CDC7 O00311 1/20 0.35
ROCK2 O75116 1/20 0.35
MAP4K4 O95819 1/20 0.35
PIM1 P11309 1/20 0.35
PRKACA P17612 1/20 0.35
CDK2 P24941 1/20 0.35
GSK3B P49841 1/20 0.35
HIPK2 Q9H2X6 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
BACE1 P56817 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3776705 0.99 INPPL1 (0.36) INPPL1CYP11B1CYP11B2CHRNB2CHRNB1
SCHEMBL3141790 0.86 CHRNB2 (0.48) INPPL1CYP11B1CYP11B2CHRNB2CHRNB1
SCHEMBL3150922 0.85 CHRNB1 (0.49) INPPL1CYP11B1CYP11B2CHRNB2CHRNB1
Hydrochloric Acid SCHEMBL3773084 0.85 CHRNB2 (0.47) INPPL1CYP11B1CYP11B2CHRNB2CHRNB1
SCHEMBL3145280 0.85 CHRNB1 (0.49) INPPL1CYP11B1CYP11B2CHRNB2CHRNB1
SCHEMBL3151157 0.85 CHRNB1 (0.49) CYP11B1CYP11B2CHRNB2CHRNB1CHRNB4
SCHEMBL3147229 0.85 CHRNB2 (0.49) INPPL1CYP11B1CYP11B2CHRNB2CHRNB1
Hydrochloric Acid SCHEMBL3151937 0.84 CHRNB1 (0.48) INPPL1CYP11B1CYP11B2CHRNB2CHRNB1
SCHEMBL3145991 0.84 CYP11B1 (0.40) INPPL1CYP11B1CYP11B2CHRNB2CHRNB1
Hydrochloric Acid SCHEMBL3147131 0.84 CHRNB1 (0.48) CYP11B1CYP11B2CHRNB2CHRNB1CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed