SCHEMBL3147229

SCHEMBL3147229

CNC1(COc2cncc(-c3ccccc3)c2)CC1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.49
CHRNA4 P43681 1/20 0.49
CHRNB1 P11230 2/20 0.47
CHRNB4 P30926 2/20 0.47
CHRNA3 P32297 2/20 0.47
CHRNB3 Q05901 2/20 0.47
CYP11B1 P15538 2/20 0.39
CYP11B2 P19099 2/20 0.39
INPPL1 O15357 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3765553 0.99 CHRNB2 (0.48) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL3141790 0.88 CHRNB2 (0.48) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL3142735 0.87 S1PR1 (0.38) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL3150645 0.87 CYP11B1 (0.47) CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL3773084 0.87 CHRNB2 (0.47) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL3145280 0.87 CHRNB1 (0.49) CHRNB2CHRNB1CHRNB4CHRNA3CHRNB3
SCHEMBL3151157 0.87 CHRNB1 (0.49) CHRNB2CHRNB1CHRNB4CHRNA3CHRNB3
SCHEMBL3150922 0.87 CHRNB1 (0.49) CHRNB2CHRNB1CHRNB4CHRNA3CHRNB3
SCHEMBL3147306 0.86 INPPL1 (0.43) CHRNB2CHRNB1CHRNB4CHRNA3CHRNB3
SCHEMBL3146014 0.86 CHRNB1 (0.52) CHRNB2CHRNB1CHRNB4CHRNA3CHRNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed