SCHEMBL3154271

SCHEMBL3154271

CCN(CC)c1cccc(ON(c2ccccc2)S(=O)(=O)c2ccc(C(=O)NC3CCC(CCN4CCCC4)CC3)cc2)c1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 16/20 0.44
DRD3 P35462 16/20 0.44
HTR2A P28223 9/20 0.44
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3149102 0.91 DRD2 (0.51) DRD2DRD3HTR2ALMNASMN1; SMN2
SCHEMBL3143699 0.86 DRD2 (0.47) DRD2DRD3HTR2ALMNASMN1; SMN2
SCHEMBL3145983 0.86 DRD2 (0.50) DRD2DRD3HTR2A
SCHEMBL3157844 0.85 DRD2 (0.47) DRD2DRD3HTR2ALMNASMN1; SMN2
SCHEMBL3149086 0.84 CA12 (0.49) LMNASMN1; SMN2
SCHEMBL3154260 0.83 RAB9A (0.44) DRD2DRD3HTR2A
SCHEMBL3154254 0.83 RAB9A (0.44) DRD2DRD3HTR2A
SCHEMBL3044402 0.83 DRD2 (0.43) DRD2DRD3HTR2A
SCHEMBL3149321 0.82 KMT2A (0.47) DRD2DRD3HTR2ALMNASMN1; SMN2
SCHEMBL3148961 0.81 DRD3 (0.46) DRD2DRD3HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074083-B1 NEW SULFONAMIDE DERIVATIVES AS BRADYKININ ANTAGONISTS RICHTER GEDEON NYRT (HU) 2013-06-19 EP disclosed
US-20100075978-A1 SULFONAMIDE DERIVATIVES AS BRADYKININ ANTAGONISTS RICHTER GEDEON NYRT. (HU) 2010-03-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100075978-A1 SULFONAMIDE DERIVATIVES AS BRADYKININ ANTAGONISTS BDKRB1, BDKRB2, TRPV1 DRD2 424/4885DRD3 467/4885HTR2A 985/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.